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Found 230 with Last Name = 'sato' and Initial = 'i'
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394470(CHEMBL2160099)
Affinity DataIC50:  0.870nMAssay Description:Antagonist activity at CCR3 receptor in human eosinophils assessed as inhibition of CCL11-induced degranulation after 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297172(CHEMBL560275 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  0.980nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297171(CHEMBL551735 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells by functional inhibition curve analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297181(2-[1-(1,3-Benzodioxol-5-ylcarbonyl)piperidin-4-yli...)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394470(CHEMBL2160099)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297183(CHEMBL551738 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  1.80nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394487(CHEMBL2160111)
Affinity DataIC50:  2.40nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297177(CHEMBL561535 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  3.30nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297182(2-[1-(3,4-Dimethoxybenzoyl)piperidin-4-ylidene]-N-...)
Affinity DataIC50:  3.60nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297190(2-(1-Benzoylpiperidin-4-ylidene)-N-{(3R)-1-[(6-flu...)
Affinity DataIC50:  4.40nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297188(2-[1-(2-Fluorobenzoyl)piperidin-4-ylidene]-N-{(3R)...)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387669(CHEMBL2058071)
Affinity DataIC50:  4.90nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297180(CHEMBL556916 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297179(CHEMBL562923 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  5.10nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297185(CHEMBL556227 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  5.10nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297184(CHEMBL557118 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  5.80nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297174(2-[1-(4-Fluoro-2-hydroxybenzoyl)piperidin-4-yliden...)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297173(2-[1-(4-Chloro-2-hydroxybenzoyl)piperidin-4-yliden...)
Affinity DataIC50:  7.5nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387649(CHEMBL2057751)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297171(CHEMBL551735 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  8.40nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394482(CHEMBL2159867)
Affinity DataIC50:  9.90nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394481(CHEMBL2159868)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264210(2-(Azepan-1-ylcarbonyl)-N-{(3-exo)-8-[(6-fluoro-2-...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at CCR3 receptor expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium influx by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297187((R)-2-(1-(3-fluorobenzoyl)piperidin-4-ylidene)-N-(...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387664(CHEMBL2057766)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387661(CHEMBL2057763)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264161(CHEMBL488929 | N-{(3-exo)-8-[(6-Fluoro-2-naphthyl)...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at CCR3 receptor expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium influx by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394486(CHEMBL2159863)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297176(CHEMBL562574 | N-{(3R)-1-[(6-Fluoro-2-naphthyl)met...)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Meiji Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM16034(1-N-[(2S,3R)-4-(cyclopropylamino)-3-hydroxy-1-phen...)
Affinity DataIC50:  15nMAssay Description:Inhibition of BACE1 (unknown origin) using Rh-EVNNLDAEFK fluorogenic peptide as substrate incubated for 3 hrs by FRET assayMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Meiji Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM16034(1-N-[(2S,3R)-4-(cyclopropylamino)-3-hydroxy-1-phen...)
Affinity DataIC50:  15nMAssay Description:Inhibition of BACE1 (unknown origin) using Rh-EVNNLDAEFK-Quencher substrate incubated for 3 hrs by FRET assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387654(CHEMBL2057756)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50264142(Biphenyl-2-carboxylic acid [(1R,5R)-8-(6-fluoro-na...)
Affinity DataIC50:  20nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387642(CHEMBL2057491)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264142(Biphenyl-2-carboxylic acid [(1R,5R)-8-(6-fluoro-na...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CCR3 receptor expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium influx by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50375019(CHEMBL258996)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CCR3 expressed in B300-19 cells assessed as inhibition of eotaxin-induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50375019(CHEMBL258996)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CCR3 expressed in B300-19 cells assessed as inhibition of eotaxin-induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264142(Biphenyl-2-carboxylic acid [(1R,5R)-8-(6-fluoro-na...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264142(Biphenyl-2-carboxylic acid [(1R,5R)-8-(6-fluoro-na...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CCR3 receptor expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium influx by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50297186(2-[1-(4-Fluorobenzoyl)piperidin-4-ylidene]-N-{(3R)...)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394479(CHEMBL2160097)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264212(CHEMBL519042 | N-{(3-exo)-8-[(6-Fluoro-2-naphthyl)...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at human CCR3 expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264157(CHEMBL519750 | N-{(3-exo)-8-[(6-Fluoro-2-naphthyl)...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at CCR3 receptor expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium influx by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264212(CHEMBL519042 | N-{(3-exo)-8-[(6-Fluoro-2-naphthyl)...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at CCR3 receptor expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium influx by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394480(CHEMBL2159869)
Affinity DataIC50:  24nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394488(CHEMBL2160110)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394477(CHEMBL2160100)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387665(CHEMBL2058070)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50264144(CHEMBL524113 | N-{(3-exo)-8-[(6-Fluoro-2-naphthyl)...)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at CCR3 receptor expressed in mouse B300-19 cells assessed as inhibition of eotaxin-induced calcium influx by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50387667(CHEMBL2058073)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human CCR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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