Affinity DataKi: 0.0230nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:In vitro binding affinity at opioid receptor kappa 1 was determined in human CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:In vitro binding affinity at opioid receptor kappa 1 was determined in human CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:In vitro binding affinity at opioid receptor kappa 1 was determined in human CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:In vitro binding affinity at opioid receptor kappa 1 was determined in human CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:In vitro binding affinity at opioid receptor kappa 1 was determined in human CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding affinity at opioid receptor kappa 1 was determined in human CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 0.920nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 1.18nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.25nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity at opioid receptor kappa 1 was determined in human CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 2.14nMAssay Description:Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 2.46nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.92nMAssay Description:Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.14nMAssay Description:Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.67nMAssay Description:Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair
Affinity DataKi: 6.55nMAssay Description:In vitro binding affinity at opioid receptor mu 1 was determined in C6 rat glioma cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 6.55nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 10.2nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10.3nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13.3nMAssay Description:Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 25.2nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 33.2nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 33.8nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 40.9nMAssay Description:In vitro binding affinity at opioid receptor delta 1 was determined in C6 rat glioma cells using [3H]Ile5,6 deltorphin IIMore data for this Ligand-Target Pair