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Found 901 with Last Name = 'schmeck' and Initial = 'c'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM466529(2-{[5-Acetyl-1-(2-chlorophenyl)-1H-1,2,4-triazol-3...)
Affinity DataIC50:  0.5nMAssay Description:The identification of agonists and antagonists of the V1a and V2 vasopressin receptors from humans, rats and dogs as well as the quantification of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM190302(US9180120, 6)
Affinity DataIC50:  1nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtitre plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V1a receptor(Homo sapiens (Human))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM190298(US9180120, 2)
Affinity DataIC50:  1nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtitre plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V1a receptor(Homo sapiens (Human))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM466533(US10800746, Example WO 2011/104322 56)
Affinity DataIC50:  1.30nMAssay Description:The identification of agonists and antagonists of the V1a and V2 vasopressin receptors from humans, rats and dogs as well as the quantification of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM192452(US9187466, 50 | US9687476, 50)
Affinity DataIC50:  1.40nMT: 2°CAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtiter plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM192452(US9187466, 50 | US9687476, 50)
Affinity DataIC50:  1.40nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtiter plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM192451(US9187466, 49 | US9687476, 49)
Affinity DataIC50:  1.5nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtiter plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM192451(US9187466, 49 | US9687476, 49)
Affinity DataIC50:  1.5nMT: 2°CAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtiter plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531482(6-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(cy...)
Affinity DataIC50: <1.60nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531920(4-[5-{[6-(3,5-dimethyl-1H-pyrazol-1-yl)pyrimidin-4...)
Affinity DataIC50:  1.60nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531586(US11208400, Example 219 | ethyl 1-(6-{[1-(4-cyanop...)
Affinity DataIC50: <1.60nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531488(N-[1-(cyclopropylmethyl)-4-ethyl-3-(4-fluorophenyl...)
Affinity DataIC50: <1.60nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531919(4-[5-({6-[5-(difluoromethyl)-3-methyl-1H-pyrazol-1...)
Affinity DataIC50:  1.90nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531777(4-[3-({6-[5-(difluoromethyl)-3-methyl-1H-pyrazol-1...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM192449(US9187466, 32 | US9687476, 32)
Affinity DataIC50:  2nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtiter plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531622(4-(3-{[6-(4-bromo-3,5-dimethyl-1H-pyrazol-1-yl)pyr...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531709((�)-4-{1-(cyclopropylmethyl)-5-[(6-{4-[1-et...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531428(US11208400, Example 356 | US11208400, Example 61 |...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531523(US11208400, Example 156 | ethyl 1-(6-{[3-(4-cyanop...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531528(4-[1-(cyclopropylmethyl)-5-{[6-(3,5-dimethyl-1H-py...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531563(4-(3-{[6-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)py...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531580(US11208400, Example 213 | ethyl 1-(6-{[3-(4-cyanop...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531584(4-[3-({6-[5-(difluoromethyl)-3-methyl-1H-pyrazol-1...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531598(4-[1-(cyclopropylmethyl)-4-methyl-5-{[6-(3-methyl-...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531831(4-[1-(cyclopropylmethyl)-5-{[6-(4-methoxy-3,5-dime...)
Affinity DataIC50:  2nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM190348(US9180120, 52)
Affinity DataIC50:  2nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtitre plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM192449(US9187466, 32 | US9687476, 32)
Affinity DataIC50:  2nMT: 2°CAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtiter plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM190343(US9180120, 47)
Affinity DataIC50:  2nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtitre plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM466527(2-{[5-Acetyl-1-(3-chlorophenyl)-1H-1,2,4-triazol-3...)
Affinity DataIC50:  2.30nMAssay Description:The identification of agonists and antagonists of the V1a and V2 vasopressin receptors from humans, rats and dogs as well as the quantification of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM466531(5-(4-Chlorophenyl)-2-({1-(3-chlorophenyl)-5-[(1S,R...)
Affinity DataIC50:  2.80nMAssay Description:The identification of agonists and antagonists of the V1a and V2 vasopressin receptors from humans, rats and dogs as well as the quantification of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531864(1-(6-{[1-(cyclopropylmethyl)-3-(4-fluorophenyl)-4-...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531773(6-(4-bromo-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(cyc...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM190338(US9180120, 42)
Affinity DataIC50:  3nMAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtitre plates an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50312718(CHEMBL479527 | torcetrapib)
Affinity DataIC50:  3nMAssay Description:Inhibition of human plasma CETP assessed as [3H]cholesterol ester transfer after 18 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531602(4-[3-({6-[4-chloro-5-(difluoromethyl)-3-methyl-1H-...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531781(6-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(4-...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531837(N-[4-(difluoromethoxy)-5-(4-fluorophenyl)-1-methyl...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531864(1-(6-{[1-(cyclopropylmethyl)-3-(4-fluorophenyl)-4-...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531603(4-[3-({6-[5-(difluoromethyl)-3-methyl-1H-pyrazol-1...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531508(4-[1-(cyclopropylmethyl)-5-{[6-(3,5-dimethyl-1H-py...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531509(4-[1-(cyclopropylmethyl)-5-{(6-[5-(difluoromethyl)...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531514(US11208400, Example 147 | ethyl 1-(6-{[1-(cyclopro...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531517(4-[5-{[6-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)py...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531521(4-[5-({6-[4-chloro-5-(difluoromethyl)-3-methyl-1H-...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531532(4-[1-(cyclopropylmethyl)-5-({6-[4-(2-hydroxypropan...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531558(6-(4-bromo-3,5-dimethyl-1H-pyrazol-1-yl)-N-[4-ethy...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531562(2-[4-chloro-1-(6-{[4-ethyl-5-(4-fluorophenyl)-1-me...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531571(N-[1-(cyclopropylmethyl)-3-(4-fluorophenyl)-4-meth...)
Affinity DataIC50:  3nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent phosphate transport protein 2A(Homo sapiens)
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM531406(N-[4-chloro-3-(4-ethoxyphenyl)-1H-pyrazol-5-yl]-6-...)
Affinity DataIC50:  3.20nMAssay Description:For measuring Npt2a activity in a cell based assay, a stable CHO cell line with inducible Npt2a expression was generated. Therefore, CHO T-Rex cells ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM192468(US10800746, Example WO 2011/104322 110 | US9187466...)
Affinity DataIC50:  3.30nMT: 2°CAssay Description:On the day before the assay, the cells are plated out in culture medium (DMEM, 10% FCS, 2 mM glutamine, 10 mM HEPES) in 384-well microtiter plates an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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