Affinity DataKi: 2.5nMAssay Description:Binding affinity to heparin induced human Tau 441 at 50 pM to 500 nM after 30 minsMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
University Of Cambridge
Curated by ChEMBL
University Of Cambridge
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive inhibition of full length recombinant human GSK-3alpha expressed in baculovirus infected insect Sf9 cells using GS-2 peptide as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 8.10nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: <10nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
University Of Cambridge
Curated by ChEMBL
University Of Cambridge
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of full length recombinant human GSK-3alpha expressed in baculovirus infected insect Sf9 cells using GS-2 peptide as substrate assessed as...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory activity against aldose reductase isolated from human placentaMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair