TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hebrew University of Jerusalem
Curated by ChEMBL
Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Binding affinity of the compound to opioid receptor mu was determined in rat brain using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hebrew University of Jerusalem
Curated by ChEMBL
Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Binding affinity of the compound to opioid receptor mu was determined in rat brain using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hebrew University of Jerusalem
Curated by ChEMBL
Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Binding affinity of the compound to opioid receptor delta was determined in rat brain using [3H]-DSTBULET as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hebrew University of Jerusalem
Curated by ChEMBL
Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataKi: 629nMAssay Description:Binding affinity of the compound to opioid receptor delta was determined in rat brain using [3H]-DSTBULET as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hebrew University of Jerusalem
Curated by ChEMBL
Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataKi: 1.38E+3nMAssay Description:Binding affinity of the compound to opioid receptor mu was determined in rat brain using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hebrew University of Jerusalem
Curated by ChEMBL
Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:Binding affinity of the compound to opioid receptor delta was determined in rat brain using [3H]-DSTBULET as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 6nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 265nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:In vitro smooth muscle contraction activity in guinea pig stomach consisting of CCK/gastrin receptor subtypeMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Effective dose of the compound was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methy...More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Effective dose of the compound was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methy...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Effective dose of the compound was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methy...More data for this Ligand-Target Pair
Affinity DataEC50: 600nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Compound was evaluated for effective dose against muscular receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Compound was evaluated for effective dose against Neuronal receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair