Compile Data Set for Download or QSAR
maximum 50k data
Found 122 with Last Name = 'sheets' and Initial = 'kr'
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039087(3-(3-Fluoro-4-methoxy-phenyl)-6,7-dimethoxy-quinol...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.003-0.005More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039073(5,7-Dimethyl-3-thiophen-3-yl-quinoline | CHEMBL304...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.001-0.005More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039041(6,7-Dimethoxy-3-((E)-styryl)-quinoline | CHEMBL701...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.001-0.005More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039071(6,7-Dimethoxy-3-(4-methoxy-phenyl)-quinoline | CHE...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.001-0.015More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039082(6,7-Dimethoxy-3-thiophen-3-yl-quinoline | CHEMBL66...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.01-0.02More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039047(5-Fluoro-3-thiophen-3-yl-quinoline | CHEMBL305056)
Affinity DataIC50:  20nMAssay Description:Inhibition of isolated human PDGF receptor phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039084(3-(3-Fluoro-phenyl)-6,7-dimethoxy-quinoline | CHEM...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.015-0.025More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039069(7-Fluoro-3-thiophen-3-yl-quinoline | CHEMBL307093)
Affinity DataIC50:  25nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.004-0.025More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039037(4-(6,7-Dimethoxy-quinolin-3-yl)-phenol | CHEMBL303...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.02-0.03More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039067(5-(6,7-Dimethoxy-quinolin-3-yl)-1H-pyridin-2-one |...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.015-0.03More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039072(3-(5-Chloro-thiophen-2-yl)-6,7-dimethoxy-quinoline...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.007-0.03More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039042(5,7-Dimethoxy-3-thiophen-3-yl-quinoline | CHEMBL66...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.025-0.03More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039090(3-Cyclopent-1-enyl-6,7-dimethoxy-quinoline | CHEMB...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.02-0.04More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039094(6,7-Dimethoxy-3-phenylethynyl-quinoline | CHEMBL67...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.02-0.05More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039044(3-(4-Fluoro-phenyl)-6,7-dimethoxy-quinoline | CHEM...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.035-0.06More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039057(7-Methoxy-3-thiophen-3-yl-quinoline | CHEMBL68185)
Affinity DataIC50:  60nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.002-0.06More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039065(3-Benzyloxy-6,7-dimethoxy-quinoline | CHEMBL66932)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.04-0.07More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039075(6-Methoxy-3-thiophen-3-yl-quinoline | CHEMBL303184)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.05-0.07More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039062(6,7-Dimethoxy-3-(6-methoxy-pyridin-3-yl)-quinoline...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.008-0.07More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039056(Benzyl-(6,7-dimethoxy-quinolin-3-yl)-amine | CHEMB...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.02-0.08More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039079(6,7-Dimethoxy-3-thiophen-2-yl-quinoline | CHEMBL30...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.04-0.08More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039052(6,7-Dimethoxy-3-[(E)-2-(4-methoxy-phenyl)-vinyl]-q...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.03-0.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039058(6,7-Dimethoxy-3-(4-nitro-phenyl)-quinoline | CHEMB...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.07-0.15More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039054(6,7-Dimethoxy-3-phenyl-quinoline | CHEMBL66063)
Affinity DataIC50:  150nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.07-0.15More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039053(3-((E)-Styryl)-quinoline | CHEMBL65858)
Affinity DataIC50:  200nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.1-0.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039086(3-(3,4-Difluoro-phenyl)-6,7-dimethoxy-quinoline | ...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.09-0.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039055(4-(6,7-Dimethoxy-quinolin-3-yl)-benzoic acid ethyl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.1-0.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039081(3-Thiophen-3-yl-quinoline | CHEMBL304310)
Affinity DataIC50:  250nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.2-0.25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039061(6,7-Dimethoxy-3-(5-methoxy-thiophen-2-yl)-quinolin...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.1-0.25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039043(3-(3,5-Difluoro-4-methoxy-phenyl)-6,7-dimethoxy-qu...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.2-0.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039093(6,7-Dimethoxy-3-(4-methoxy-3-methyl-phenyl)-quinol...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.1-0.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039070(6,7-Dimethoxy-3-(4-methoxy-3-nitro-phenyl)-quinoli...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.15-0.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039076(3-Cyclopentyl-6,7-dimethoxy-quinoline | CHEMBL6678...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.1-0.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039033(3-Pyridin-3-yl-quinoline-6,7-diol | CHEMBL63356)
Affinity DataIC50:  500nMAssay Description:Concentration required to inhibit phosphorylation of isolated human epidermal growth factor tyrosine kinase receptor by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039049(3-(2-Cyclohexyl-ethyl)-6,7-dimethoxy-quinoline | C...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.3-0.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039066(7-Thiophen-3-yl-[1,3]dioxolo[4,5-g]quinoline | CHE...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.2-0.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039038(3-(1H-Indol-3-yl)-6,7-dimethoxy-quinoline | CHEMBL...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.1-0.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039091((Z)-3-(3,4-Dimethoxy-phenyl)-2-pyridin-3-yl-acrylo...)
Affinity DataIC50:  700nMAssay Description:Concentration required to inhibit phosphorylation of isolated human epidermal growth factor tyrosine kinase receptor by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039050(6,7-Dimethoxy-3-pyridin-3-yl-quinoline | CHEMBL304...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.1-0.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039051(6,7-Dimethoxy-3-[2-(4-methoxy-phenyl)-ethyl]-quino...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.2-0.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039078(3-(3-Chloro-thiophen-2-yl)-6,7-dimethoxy-quinoline...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of isolated human PDGF receptor phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039040(3-Cyclohexylethynyl-6,7-dimethoxy-quinoline | CHEM...)
Affinity DataIC50:  1.00E+3nMAssay Description:Concentration required to inhibit phosphorylation of isolated human PDGF receptor by 50%; 0.3-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039080(6,7-Dimethoxy-3-p-tolyl-quinoline | CHEMBL67219)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.5-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039095(6,7-Dimethoxy-3-(2-methoxy-phenyl)-quinoline | CHE...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of isolated human PDGF receptor phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039039(6,7-Dichloro-3-thiophen-3-yl-quinoline | CHEMBL667...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 1-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039088(6,7-Dimethoxy-3-(3-methoxy-phenyl)-quinoline | CHE...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 1-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039091((Z)-3-(3,4-Dimethoxy-phenyl)-2-pyridin-3-yl-acrylo...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.5-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039085(6,7-Difluoro-3-thiophen-3-yl-quinoline | CHEMBL681...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 2-4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039077(4-(6,7-Dimethoxy-quinolin-3-yl)-benzoic acid | CHE...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 0.7-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50039074(3-(3,4-Dichloro-phenyl)-6,7-dimethoxy-quinoline | ...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human PDGF receptor phosphorylation; 1-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 122 total ) | Next | Last >>
Jump to: