Compile Data Set for Download or QSAR
maximum 50k data
Found 1342 with Last Name = 'silvian' and Initial = 'l'
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50548191(CHEMBL4793665)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of human HGK using MBP as substrate assessed as residual activity by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263757((E)-3-(4-(3-(1-isopropylpiperidin-4-ylamino)phenyl...)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50264878((cis)-4-((2-(4-((E)-3-morpholino-3-oxoprop-1-enyl)...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263657((cis)-4-(3-(4-((E)-3-morpholino-3-oxoprop-1-enyl)-...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263755((E)-3-(4-(3-(1-methylpiperidin-4-ylamino)phenylthi...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50264880((trans)-4-((2-(4-((E)-3-morpholino-3-oxoprop-1-eny...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263805((E)-1-morpholino-3-(4-(3-(1-propylpiperidin-4-ylam...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263806((E)-3-(4-(3-(8-methyl-8-azabicyclo[3.2.1]octan-3-y...)
Affinity DataIC50:  0.940nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50610140(CHEMBL5266817)
Affinity DataIC50: <1nMAssay Description:Inhibition of unphosphorylated BTK (unknown origin) in the presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042868(CHEMBL3354518)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50522686(CHEMBL4564973)
Affinity DataIC50:  1nMAssay Description:Reversible inhibition of recombinant full-length N-terminal 6-His-tagged human BTK expressed in baculovirus infected Sf21 insect cells using fluoresc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50588044(CHEMBL5176609)
Affinity DataIC50:  1nMAssay Description:Inhibition of BTK (unknown origin) incubated 30 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50352206(CHEMBL1825089)
Affinity DataIC50:  1nMAssay Description:Inhibition of CYP2C9 using a fluorescent probe 7-methoxy-4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50610140(CHEMBL5266817)
Affinity DataIC50: <1nMAssay Description:Inhibition of unphosphorylated BTK (unknown origin) in the presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042867(CHEMBL3354517)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042866(CHEMBL3354516)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042864(CHEMBL3354514)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042863(CHEMBL3354513)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042871(CHEMBL3354521)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042868(CHEMBL3354518)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042868(CHEMBL3354518)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042863(CHEMBL3354513)
Affinity DataIC50:  1nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263756((E)-3-(4-(3-(1-ethylpiperidin-4-ylamino)phenylthio...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263711((E)-1-morpholino-3-(4-(3-(piperidin-4-ylamino)phen...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263710((trans)-4-((3-(4-((E)-3-morpholino-3-oxoprop-1-eny...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM31093(4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-py...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50379503(CHEMBL2012415)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263548((E)-3-(4-(3-aminophenylthio)-2,3-bis(trifluorometh...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50265320((trans)-4-(2-(4-((E)-3-morpholino-3-oxoprop-1-enyl...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50610128(CHEMBL5284310)
Affinity DataIC50:  2nMAssay Description:Inhibition of unphosphorylated BTK (unknown origin) in the presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50610136(CHEMBL5274179)
Affinity DataIC50:  2nMAssay Description:Inhibition of unphosphorylated BTK (unknown origin) in the presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50265147((E)-1-morpholino-3-(4-(2-(piperidin-4-yloxy)phenyl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042867(CHEMBL3354517)
Affinity DataIC50:  2nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50042861(CHEMBL3354511)
Affinity DataIC50:  2nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50610137(CHEMBL5269111)
Affinity DataIC50:  2nMAssay Description:Inhibition of unphosphorylated BTK (unknown origin) in the presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50610139(CHEMBL5287698)
Affinity DataIC50:  2nMAssay Description:Inhibition of unphosphorylated BTK (unknown origin) in the presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50384165(CHEMBL2029908)
Affinity DataIC50:  2nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50384166(CHEMBL2029909)
Affinity DataIC50:  2nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50384167(CHEMBL2029910)
Affinity DataIC50:  2nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50384168(CHEMBL2029911)
Affinity DataIC50:  2nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50384169(CHEMBL2029912)
Affinity DataIC50:  2nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50384171(CHEMBL2029914)
Affinity DataIC50:  2nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50379494(CHEMBL2012406)
Affinity DataIC50:  2nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50265190((E)-1-morpholino-3-(4-(3-(tetrahydro-2H-thiopyran-...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50263656((trans)-4-(3-(4-((E)-3-morpholino-3-oxoprop-1-enyl...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50264778((E)-1-morpholino-3-(4-(2-(pyridin-3-ylmethoxy)phen...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
TargetIntegrin alpha-L(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50265149((E)-1-morpholino-3-(4-(2-(tetrahydro-2H-pyran-4-yl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of recombinant LFA1/ICAM1-IG interaction (unknown origin) by time-resolved fluorimetry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50610138(CHEMBL5268773)
Affinity DataIC50:  3nMAssay Description:Inhibition of unphosphorylated BTK (unknown origin) in the presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 3(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50548192(CHEMBL4749141)
Affinity DataIC50:  3nMAssay Description:Inhibition of GLK (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50352202(CHEMBL1825101)
Affinity DataIC50:  3nMAssay Description:Inhibition of CDK1/Cyclin B assessed as phosphorylation of Z-lyte Peptide at 0.017 to 30 nM by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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