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Found 184 with Last Name = 'snell' and Initial = 'cr'
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370083(CHEMBL1907651)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370077(CHEMBL1907652)
Affinity DataKi:  0.310nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409120(CHEMBL2112044 | CHEMBL2112937)
Affinity DataKi:  0.5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50113263((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409120(CHEMBL2112044 | CHEMBL2112937)
Affinity DataKi:  0.600nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50113263((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409527(CHEMBL2112283)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409529(CHEMBL2112221)
Affinity DataKi:  1.47nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085685(4-benzhydrylamino(thioxo)methylhydrazine-3-nitrobe...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409528(CHEMBL2112220)
Affinity DataKi:  2.79nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085684(4-benzhydrylamino(thioxo)methylhydrazine-3-nitro-1...)
Affinity DataKi:  4nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370080(CHEMBL1907656)
Affinity DataKi:  4.67nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370081(CHEMBL1907654)
Affinity DataKi:  5.46nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370078(CHEMBL1907653)
Affinity DataKi:  7.30nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409527(CHEMBL2112283)
Affinity DataKi:  10.7nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370080(CHEMBL1907656)
Affinity DataKi:  14.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370081(CHEMBL1907654)
Affinity DataKi:  34.1nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085698(CHEMBL164636 | benzhydrylamino-2-nitrobenzylhydraz...)
Affinity DataKi:  38nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409529(CHEMBL2112221)
Affinity DataKi:  64.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370077(CHEMBL1907652)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370083(CHEMBL1907651)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085696(1N,1N-di(3-dimethylaminopropyl)-4-benzhydrylamino(...)
Affinity DataKi:  148nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409528(CHEMBL2112220)
Affinity DataKi:  176nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50113264(1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzen...)
Affinity DataKi:  237nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409530(CHEMBL2112219)
Affinity DataKi:  253nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370082(CHEMBL1907655)
Affinity DataKi:  299nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085689(1N-benzyl-4-benzylamino(thioxo)methylhydrazine-3-n...)
Affinity DataKi:  310nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085692(2-{4-[2-furylmethylamino(thioxo)methylhydrazine]-3...)
Affinity DataKi:  540nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370084(CHEMBL1907657)
Affinity DataKi:  645nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50370082(CHEMBL1907655)
Affinity DataKi:  654nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50113263((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...)
Affinity DataKi:  772nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50113263((S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobe...)
Affinity DataKi:  1.43E+3nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085694(CHEMBL163956 | benzylamino-2-nitrobenzylhydrazinem...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085690(1-Benzyl-3-(2-nitro-benzyl)-thiourea | CHEMBL16524...)
Affinity DataKi:  7.10E+3nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085695(CHEMBL164551 | N-Benzyl-3-nitro-4-[N'-(3-phenyl-th...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085697(1-Benzyl-3-(2-nitro-benzyl)-urea | CHEMBL165238)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085691(CHEMBL350109 | N-Benzyl-2-(4-benzylsulfamoyl-2-nit...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085686(2-benzylamino(thioxo)methylhydrazinebenzoic acid |...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085688(CHEMBL164914 | benzylamino-3-nitrobenzylhydrazinem...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085687(CHEMBL164968 | phenyl-hydrazine-1-benzylamino-1-me...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409528(CHEMBL2112220)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of Bradykinin receptor B2-mediated contractions of rat uterus smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50252500(6-(4-chlorobenzyl)-7-(3,3-dimethylbutyl)-7H-pyrrol...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant cathepsin S by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50251889(4-((2-cyano-7-(2-cyclohexylethyl)-7H-pyrrolo[2,3-d...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant cathepsin S by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50409527(CHEMBL2112283)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of Bradykinin receptor B2-mediated contractions of rat uterus smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataIC50:  2.90nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50252502(6-(4-chlorobenzyl)-7-(cyclohexylmethyl)-7H-pyrrolo...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50251887(3-(3-((2-cyano-7-(2-cyclohexylethyl)-7H-pyrrolo[2,...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant cathepsin S by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50252656(7-(2-cyclohexylethyl)-6-((pyridin-4-yloxy)methyl)-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant cathepsin S by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50252543(6-(4-chlorobenzyl)-7-(2-cyclopentylethyl)-7H-pyrro...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant cathepsin S by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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