Compile Data Set for Download or QSAR
maximum 50k data
Found 201 with Last Name = 'stirnberg' and Initial = 'm'
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324477(Benzylsulfonyl-D-cyclohexylalanyl-proline-(4-amidi...)
Affinity DataKi:  0.102nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324478(Benzylsulfonyl-D-cyclohexylalanyl-proline-(2-amino...)
Affinity DataKi:  0.108nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324476(Benzylsulfonyl-D-arginyl-proline-(2-aminomethyl-5-...)
Affinity DataKi:  1nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324475(Benzylsulfonyl-D-argininyl-proline-(4-amidinobenzy...)
Affinity DataKi:  1.94nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324475(Benzylsulfonyl-D-argininyl-proline-(4-amidinobenzy...)
Affinity DataKi:  55nMAssay Description:Inhibition of human recombinant matriptase catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324475(Benzylsulfonyl-D-argininyl-proline-(4-amidinobenzy...)
Affinity DataKi:  170nMAssay Description:Inhibition of human purified matriptase 2 catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324475(Benzylsulfonyl-D-argininyl-proline-(4-amidinobenzy...)
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant matriptase 2 expressed in HEK293 cells in conditioned medium after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189306(CHEMBL3594083)
Affinity DataKi:  192nMAssay Description:Inhibition of human trypsin using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324476(Benzylsulfonyl-D-arginyl-proline-(2-aminomethyl-5-...)
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant matriptase catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189311(4,4''-(1,2-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  221nMAssay Description:Inhibition of human trypsin using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189307(CHEMBL3594082)
Affinity DataKi:  244nMAssay Description:Inhibition of human trypsin using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189311(4,4''-(1,2-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  279nMAssay Description:Inhibition of human thrombin using Cbz-Gly-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324477(Benzylsulfonyl-D-cyclohexylalanyl-proline-(4-amidi...)
Affinity DataKi:  290nMAssay Description:Inhibition of human recombinant matriptase 2 expressed in HEK293 cells in conditioned medium after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189310(4,4''-(1,4-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  316nMAssay Description:Inhibition of human trypsin using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189306(CHEMBL3594083)
Affinity DataKi:  317nMAssay Description:Inhibition of human thrombin using Cbz-Gly-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bos taurus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189310(4,4''-(1,4-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  327nMAssay Description:Inhibition of bovine factor 10a using Boc-Ile-Glu-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bos taurus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189307(CHEMBL3594082)
Affinity DataKi:  391nMAssay Description:Inhibition of bovine factor 10a using Boc-Ile-Glu-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189308(CHEMBL269032)
Affinity DataKi:  397nMAssay Description:Inhibition of human matriptase using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324477(Benzylsulfonyl-D-cyclohexylalanyl-proline-(4-amidi...)
Affinity DataKi:  460nMAssay Description:Inhibition of human purified matriptase 2 catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189305(CHEMBL3828410)
Affinity DataKi:  492nMAssay Description:Inhibition of human matriptase using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189307(CHEMBL3594082)
Affinity DataKi:  499nMAssay Description:Inhibition of human thrombin using Cbz-Gly-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189309(CHEMBL9126)
Affinity DataKi:  513nMAssay Description:Inhibition of human trypsin using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189306(CHEMBL3594083)
Affinity DataKi:  526nMAssay Description:Inhibition of human matriptase using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50394250(CHEMBL2159280)
Affinity DataKi:  530nMAssay Description:Inhibition of human thrombin using fluorogenic Cbz-Gly-Gly-Arg-NH-Mec as substrate measured over 400 secs by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189307(CHEMBL3594082)
Affinity DataKi:  558nMAssay Description:Inhibition of human matriptase using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189309(CHEMBL9126)
Affinity DataKi:  719nMAssay Description:Inhibition of human matriptase using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324477(Benzylsulfonyl-D-cyclohexylalanyl-proline-(4-amidi...)
Affinity DataKi:  770nMAssay Description:Inhibition of human recombinant matriptase catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189310(4,4''-(1,4-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  816nMAssay Description:Inhibition of human matriptase using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50394254(CHEMBL2159276)
Affinity DataKi:  930nMAssay Description:Inhibition of human thrombin using fluorogenic Cbz-Gly-Gly-Arg-NH-Mec as substrate measured over 400 secs by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189310(4,4''-(1,4-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of human thrombin using Cbz-Gly-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189309(CHEMBL9126)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of human matriptase-2 transfected in HEK cells using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bos taurus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189306(CHEMBL3594083)
Affinity DataKi:  1.29E+3nMAssay Description:Inhibition of bovine factor 10a using Boc-Ile-Glu-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189305(CHEMBL3828410)
Affinity DataKi:  1.42E+3nMAssay Description:Inhibition of human trypsin using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189306(CHEMBL3594083)
Affinity DataKi:  1.64E+3nMAssay Description:Inhibition of human matriptase-2 transfected in HEK cells using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189308(CHEMBL269032)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human trypsin using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50286441((S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylami...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human recombinant matriptase catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50324478(Benzylsulfonyl-D-cyclohexylalanyl-proline-(2-amino...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of human recombinant matriptase catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189311(4,4''-(1,2-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  2.28E+3nMAssay Description:Inhibition of human matriptase using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50394252(CHEMBL2159278)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of human thrombin using fluorogenic Cbz-Gly-Gly-Arg-NH-Mec as substrate measured over 400 secs by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50286441((S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylami...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of human recombinant matriptase 2 expressed in HEK293 cells in conditioned medium after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189310(4,4''-(1,4-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of bovine thrombin using BANA/BPVANA as substrate after 15 to 40 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189307(CHEMBL3594082)
Affinity DataKi:  3.68E+3nMAssay Description:Inhibition of human matriptase-2 transfected in HEK cells using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50394293(CHEMBL2159394)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of human thrombin using fluorogenic Cbz-Gly-Gly-Arg-NH-Mec as substrate measured over 400 secs by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50286441((S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylami...)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of human purified matriptase 2 catalytic domain expressed in HEK293 cells after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189308(CHEMBL269032)
Affinity DataKi:  4.39E+3nMAssay Description:Inhibition of human matriptase-2 transfected in HEK cells using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50394258(CHEMBL2159272)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of human thrombin using fluorogenic Cbz-Gly-Gly-Arg-NH-Mec as substrate measured over 400 secs by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189311(4,4''-(1,2-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of human matriptase-2 transfected in HEK cells using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189308(CHEMBL269032)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of human thrombin using Cbz-Gly-Gly-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50189310(4,4''-(1,4-Phenylenebis(Methylene))Bis(Oxy)Dibenzi...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of human matriptase-2 transfected in HEK cells using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50394288(CHEMBL2159282)
Affinity DataKi:  5.82E+3nMAssay Description:Inhibition of human thrombin using fluorogenic Cbz-Gly-Gly-Arg-NH-Mec as substrate measured over 400 secs by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 201 total ) | Next | Last >>
Jump to: