Compile Data Set for Download or QSAR
maximum 50k data
Found 2616 with Last Name = 'stocks' and Initial = 'mj'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  0.0794nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetP2Y purinoceptor 12(Homo sapiens (Human))TBA
LigandPNGBDBM50167271(CHEMBL3798413)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-2-MeS-ADP from human P2Y12 assessed as inhibition constant incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Kalvista Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM408717( N-[(3-fluoro-4-methoxypyridin-2-yl)methyl]-3-(met...)
Affinity DataKi:  3nMAssay Description:Reversible inhibition of human plasma kallikrein assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429537(CHEMBL2333770)
Affinity DataKi:  6nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429541(CHEMBL2333766)
Affinity DataKi:  7nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429548(CHEMBL2333759)
Affinity DataKi:  18nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429538(CHEMBL2333767)
Affinity DataKi:  20nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))TBA
LigandPNGBDBM50268964(CHEMBL502519 | Sodium 1-Amino-4-[4-phenylamino-3-c...)
Affinity DataKi:  21nMAssay Description:Antagonist activity at human P2Y12 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  22nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(2-(4-(2-(5,5-difluoro-7-(thiophen-2-yl)-5H-4-lambda4,5-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazab...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429546(CHEMBL2333761)
Affinity DataKi:  28nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373303(CHEMBL256141)
Affinity DataKi:  30nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429547(CHEMBL2333760)
Affinity DataKi:  33nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  35nMAssay Description:Displacement of N-(2-(3-((7-Chloro-4-(1-methyl-2-oxo-4-thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-4H-benzo[5,6]cyclohepta[1,2-d]thiazol-2-yl)-amino)pro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  42nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429567(CHEMBL2333776)
Affinity DataKi:  47nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  48nMAssay Description:Displacement of N-(2-(2-(2-(3-((7-Chloro-4-(1-methyl-2-oxo-4-thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-4H-benzo[5,6]cyclohepta[1,2-d]thiazol-2-yl)amin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429561(CHEMBL2333353)
Affinity DataKi:  48nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429562(CHEMBL2333352)
Affinity DataKi:  69nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373324(CHEMBL258406)
Affinity DataKi:  70nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429569(CHEMBL2333774)
Affinity DataKi:  75nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429545(CHEMBL2333762)
Affinity DataKi:  77nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))TBA
LigandPNGBDBM50614414(CHEMBL5271821)
Affinity DataKi:  80nMAssay Description:Antagonist activity at human P2Y14 expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271600(CHEMBL4086462)
Affinity DataKi:  83nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate--CoA ligase(Pseudomonas aeruginosa (Gram- Bacteria))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50324670(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKi:  88nMAssay Description:Inhibition of recombinant Pseudomonas aeruginosa PqsA assessed as decrease in formation of anthranilyl-CoA by spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373323(CHEMBL255306)
Affinity DataKi:  90nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAnthranilate--CoA ligase(Pseudomonas aeruginosa (Gram- Bacteria))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50465699(CHEMBL377483)
Affinity DataKi:  109nMAssay Description:Inhibition of recombinant Pseudomonas aeruginosa PqsA assessed as decrease in formation of anthranilyl-CoA by spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271596(CHEMBL4128126)
Affinity DataKi:  129nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271589(CHEMBL4128024)
Affinity DataKi:  145nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))TBA
LigandPNGBDBM50343128(2-(benzo[d][1,3]dioxol-5-yl)-N-(3-ethylphenyl)-4-o...)
Affinity DataKi:  160nMAssay Description:Antagonist activity at human recombinant P2Y14 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429568(CHEMBL2333775)
Affinity DataKi:  171nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429544(CHEMBL2333763)
Affinity DataKi:  172nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429540(CHEMBL2333768)
Affinity DataKi:  175nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271599(CHEMBL4128208)
Affinity DataKi:  275nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429559(CHEMBL2333355)
Affinity DataKi:  313nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271569(CHEMBL4128318)
Affinity DataKi:  398nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  501nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  501nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429565(CHEMBL2333349)
Affinity DataKi:  607nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  631nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271597(CHEMBL4127983)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429549(CHEMBL2333758)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50205417(CHEMBL220200 | UTP-gamma-S)
Affinity DataKi:  3.47E+3nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429539(CHEMBL2333769)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429551(CHEMBL2333757)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429550(CHEMBL2331579)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429542(CHEMBL2333765)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429543(CHEMBL2333764)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429566(CHEMBL2333348)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [beta-33p]-2-MeS-ADP from human P2Y1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271598(CHEMBL4128059)
Affinity DataKi:  5.25E+3nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373301(CHEMBL256944)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human P2Y1 assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Displayed 1 to 50 (of 2616 total ) | Next | Last >>
Jump to: