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Found 212 with Last Name = 'subkowski' and Initial = 't'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112996(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112986(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113007(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112985(3-(2-{[2-(3-Benzyl-ureido)-thiazole-4-carbonyl]-am...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113000(3-(2-{[2-(3-Benzyl-ureido)-oxazole-5-carbonyl]-ami...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122205((R)-4-{4-[3-(1H-Benzoimidazol-2-ylamino)-propylami...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112993((S)-2-Benzyloxycarbonylamino-3-(2-{[5-(3-benzyl-ur...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122205((R)-4-{4-[3-(1H-Benzoimidazol-2-ylamino)-propylami...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112988(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50372236(CHEMBL256672)
Affinity DataIC50:  0.700nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113013(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122219((R)-4-{4-[4-(1H-Benzoimidazol-2-ylamino)-piperidin...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122204((S)-3-{4-[4-(1H-Benzoimidazol-2-ylamino)-piperidin...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122198((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122192((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of alphaIIb-beta3 integrin binding to fibrinogen in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122195((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122227((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112987(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50411639(CHEMBL269950)
Affinity DataIC50:  1.5nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50109298(CHEMBL344162 | [5-({[4-(1H-Benzoimidazol-2-ylamino...)
Affinity DataIC50:  1.60nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113010((S)-2-Benzyloxycarbonylamino-3-(2-{[2-(3-benzyl-ur...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112990(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113015(3-(2-{[5-(3-Benzyl-ureido)-thiophene-3-carbonyl]-a...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122225((S)-2-Benzyloxycarbonylamino-3-{5-methyl-2-oxo-4-[...)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122222((R)-3-Benzyloxycarbonylamino-4-{4-[3-(1H-imidazol-...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112991((R)-2-Benzyloxycarbonylamino-3-(3-{[5-(3-benzyl-ur...)
Affinity DataIC50:  3.10nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122216((R)-3-Benzyloxycarbonylamino-4-{4-[2-(1H-imidazol-...)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113011(3-(2-{[2-(3-Benzyl-ureido)-oxazole-5-carbonyl]-ami...)
Affinity DataIC50:  3.80nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122228((S)-2-Benzyloxycarbonylamino-3-(4-{[2-(3-benzyl-ur...)
Affinity DataIC50:  4.20nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50372237(CHEMBL256673)
Affinity DataIC50:  4.20nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50411638(CHEMBL404371)
Affinity DataIC50:  4.40nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50109296((5-{[4-(1H-Benzoimidazol-2-ylamino)-benzylcarbamoy...)
Affinity DataIC50:  7nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50109296((5-{[4-(1H-Benzoimidazol-2-ylamino)-benzylcarbamoy...)
Affinity DataIC50:  7.30nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50411637(CHEMBL255952)
Affinity DataIC50:  7.40nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112999((S)-2-Benzyloxycarbonylamino-3-(2-{[5-(3-benzyl-ur...)
Affinity DataIC50:  8.90nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122218((S)-3-{4-[4-(1H-Benzoimidazol-2-yl)-piperidin-1-yl...)
Affinity DataIC50:  9.40nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122202((S)-2-Benzyloxycarbonylamino-3-{5-methyl-2-oxo-4-[...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122220((R)-4-(4-{4-[2-(1H-Benzoimidazol-2-ylamino)-ethyl]...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122198((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50411631(CHEMBL258325)
Affinity DataIC50:  10nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50411627(CHEMBL269961)
Affinity DataIC50:  11nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122229((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50109305((5-{[5-(1H-Benzoimidazol-2-ylamino)-pentylcarbamoy...)
Affinity DataIC50:  13nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50411633(CHEMBL401660)
Affinity DataIC50:  13nMAssay Description:Displacement of vitronectin from integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113002(3-(2-{[2-(3-Benzyl-ureido)-oxazole-4-carbonyl]-ami...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50109307((5-{[4-(1H-Benzoimidazol-2-ylamino)-butylcarbamoyl...)
Affinity DataIC50:  15nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122211((S)-3-(4-{4-[2-(1H-Benzoimidazol-2-ylamino)-ethyl]...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122237((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  16nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113014(3-(2-{[4-(3-Benzyl-ureido)-1-methyl-1H-pyrrole-2-c...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122214((R)-4-{4-[4-(1H-Benzoimidazol-2-ylamino)-butylamin...)
Affinity DataIC50:  17nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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