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Found 539 with Last Name = 'sunose' and Initial = 'm'
LigandPNGBDBM50387541(CHEMBL2057368)
Affinity DataIC50:  2.51nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387544(CHEMBL2057373)
Affinity DataIC50:  2.51nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387546(CHEMBL2057363)
Affinity DataIC50:  3.16nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387543(CHEMBL2057372)
Affinity DataIC50:  3.98nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642790(US11857552, Compound APPAMP-004)
Affinity DataIC50:  4.20nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642790(US11857552, Compound APPAMP-004)
Affinity DataIC50:  4.20nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642790(US11857552, Compound APPAMP-004)
Affinity DataIC50:  4.20nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50387542(CHEMBL2057371)
Affinity DataIC50:  6.31nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387541(CHEMBL2057368)
Affinity DataIC50:  6.31nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50389412(CHEMBL2064508)
Affinity DataIC50:  6.31nMAssay Description:Inhibition of PI3Kgamma by high throughput chemoproteomics binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387539(CHEMBL2057366)
Affinity DataIC50:  6.31nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401144(CHEMBL2205771)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50389431(CHEMBL2064501)
Affinity DataIC50:  7.94nMAssay Description:Inhibition of PI3Kgamma by high throughput chemoproteomics binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50389427(CHEMBL2064507)
Affinity DataIC50:  7.94nMAssay Description:Inhibition of PI3Kgamma by high throughput chemoproteomics binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387538(CHEMBL2057365)
Affinity DataIC50:  7.94nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642789(US11857552, Compound APPAMP-003)
Affinity DataIC50:  8.90nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642789(US11857552, Compound APPAMP-003)
Affinity DataIC50:  8.90nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642789(US11857552, Compound APPAMP-003)
Affinity DataIC50:  8.90nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50387540(CHEMBL2057367)
Affinity DataIC50:  10nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387536(CHEMBL2057362)
Affinity DataIC50:  12.6nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387530(CHEMBL2059910)
Affinity DataIC50:  12.6nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387544(CHEMBL2057373)
Affinity DataIC50:  12.6nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642787(US11857552, Compound APPAMP-001)
Affinity DataIC50:  13nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642787(US11857552, Compound APPAMP-001)
Affinity DataIC50:  13nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642787(US11857552, Compound APPAMP-001)
Affinity DataIC50:  13nMAssay Description:CDK7 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:CDK7/cycH/MAT1 (ProQinase, 0366-0360-4).MnCl2 (Sigma, M1787).CDKt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50401152(CHEMBL2205766)
Affinity DataIC50:  13nMAssay Description:Inhibition of CK2a1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTarget of rapamycin complex subunit LST8(Homo sapiens)
Cellzome

Curated by ChEMBL
LigandPNGBDBM50535043(CHEMBL4577549)
Affinity DataIC50:  15nMAssay Description:Inhibition of mTORC1 in HEK293T/17 cells assessed as reduction in S6RP phosphorylation at Ser-240/244 residue after 2 hrs by sandwich immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTarget of rapamycin complex 2 subunit MAPKAP1(Homo sapiens)
Cellzome

Curated by ChEMBL
LigandPNGBDBM50535043(CHEMBL4577549)
Affinity DataIC50:  15nMAssay Description:Inhibition of mTORC2 in HEK293T/17 cells assessed as reduction in Akt phosphorylation at Ser-473 residue after 2 hrs by sandwich immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387538(CHEMBL2057365)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387548(CHEMBL2059913)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387527(CHEMBL2057370)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387543(CHEMBL2057372)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50389391(CHEMBL2064512)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of PI3Kgamma by high throughput chemoproteomics binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401150(CHEMBL2205763)
Affinity DataIC50:  16nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387548(CHEMBL2059913)
Affinity DataIC50:  19.9nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401153(CHEMBL2205767)
Affinity DataIC50:  20nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401147(CHEMBL2205768)
Affinity DataIC50:  20nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401149(CHEMBL2205773)
Affinity DataIC50:  20nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Kudos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50302293(4-(1-(4,6-dimorpholino-1,3,5-triazin-2-yl)-1H-imid...)
Affinity DataIC50:  21nMAssay Description:Inhibition of mTOR kinase in human HeLa cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Carrick Therapeutics

US Patent
LigandPNGBDBM642789(US11857552, Compound APPAMP-003)
Affinity DataIC50:  22nMAssay Description:CDK9 IC50 Materials and Solutions:In addition to those mentioned above for Method 1:Human CDK9/cycK (Promega, V4104).CDKtide (SignalChem, C06-58).Ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Kudos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50302286(4-(5-(2,6-dimorpholinopyrimidin-4-yl)furan-2-yl)-2...)
Affinity DataIC50:  23nMAssay Description:Inhibition of mTOR kinase in human HeLa cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401152(CHEMBL2205766)
Affinity DataIC50:  25nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401143(CHEMBL2205774)
Affinity DataIC50:  25nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50389420(CHEMBL2064571)
Affinity DataIC50:  25nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401148(CHEMBL2205765)
Affinity DataIC50:  25nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50401146(CHEMBL2205772)
Affinity DataIC50:  25nMAssay Description:Inhibition of PIK3CgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387537(CHEMBL2057364)
Affinity DataIC50:  25.1nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387536(CHEMBL2057362)
Affinity DataIC50:  25.1nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387529(CHEMBL2059909)
Affinity DataIC50:  25.1nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50387535(CHEMBL2057361)
Affinity DataIC50:  25.1nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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