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Found 48 with Last Name = 'taghavi-moghadam' and Initial = 's'
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203110(CHEMBL3914791)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203111(CHEMBL3968023)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203043(CHEMBL3896867)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203113(CHEMBL3889816)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202837(CHEMBL3941751)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203040(CHEMBL3932774)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203048(CHEMBL3984603)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081589(CHEMBL101399 | N*4*,N*4*-Dibenzyl-6-phenyl-pteridi...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202840(CHEMBL3904763)
Affinity DataIC50:  4.54E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081585(CHEMBL100659 | N*4*,N*4*-Dibenzyl-6-(4-methoxy-phe...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203042(CHEMBL3923820)
Affinity DataIC50:  5.69E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081588(1-(2,4-Diamino-5,6,7,8-tetrahydro-pteridin-6-yl)-p...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081594(6-Phenyl-5,6,7,8-tetrahydro-pteridine-2,4-diamine ...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203044(CHEMBL3960953)
Affinity DataIC50:  9.74E+3nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202835(CHEMBL3895295)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203049(CHEMBL3904207)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203041(CHEMBL3895818)
Affinity DataIC50: <1.36E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202838(CHEBI:67605 | Eupolauridine)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081582(7-Phenyl-5,6,7,8-tetrahydro-pteridine-2,4-diamine ...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202880(CHEMBL3914880)
Affinity DataIC50:  2.82E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203046(CHEMBL3913215)
Affinity DataIC50:  2.84E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202841(CHEMBL3972163)
Affinity DataIC50:  2.88E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric-oxide synthase (NADPH)(Bos taurus)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081587(6-Decyloxymethyl-pteridine-2,4-diamine | CHEMBL986...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity against Nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081583(6-Ethoxymethyl-5,6,7,8-tetrahydro-pteridine-2,4-di...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203038(CHEMBL3975075)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081579(6-(4-Methoxy-phenyl)-4-morpholin-4-yl-pteridin-2-y...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203037(CHEMBL3890769)
Affinity DataIC50:  3.44E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203039(CHEMBL3903152)
Affinity DataIC50:  3.57E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203045(CHEMBL3915026)
Affinity DataIC50:  4.16E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081584(CHEMBL100658 | N*4*,N*4*-Diethyl-6-(4-methoxy-phen...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203047(CHEMBL3932850)
Affinity DataIC50:  4.62E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081581(3-(4-Benzoyl-phenyl)-propionic acid 2,4-diamino-pt...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202834(CHEMBL3957092)
Affinity DataIC50:  4.84E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203050(CHEMBL3984682)
Affinity DataIC50:  4.99E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081590(6-(4-Methoxy-phenyl)-4-piperidin-1-yl-pteridin-2-y...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202863(CHEMBL3896944)
Affinity DataIC50:  5.36E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081586(6-Phenyl-4-piperidin-1-yl-pteridin-2-ylamine | CHE...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202895(CHEMBL3976611)
Affinity DataIC50:  6.99E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203066(CHEMBL3904846)
Affinity DataIC50:  7.05E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081580(6-(4-Methoxy-phenyl)-N*4*,N*4*-dimethyl-pteridine-...)
Affinity DataIC50:  7.40E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081593(4-Morpholin-4-yl-6-phenyl-pteridin-2-ylamine | CHE...)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203112(CHEMBL3984838)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203051(CHEMBL3985749)
Affinity DataIC50:  1.09E+5nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202839(CHEMBL3968109)
Affinity DataIC50:  1.27E+5nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50202836(CHEMBL3894198)
Affinity DataIC50:  1.36E+5nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081591(6-Phenoxymethyl-pteridine-2,4-diamine | CHEMBL1322...)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50203067(CHEMBL3922223)
Affinity DataIC50:  2.42E+5nMAssay Description:Inhibition of human DNA topoisomerase 1 using pHOT1 as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Sus scrofa)
Julius-Maximilians University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50081592(2,4-Diamino-7,8-dihydro-6H-pteridine-5-carbaldehyd...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibitory activity against Nitric oxide synthase (derived from porcine brain cerebellum)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed