TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of DNA-PK (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: >1.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: 1.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: 2.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: 2.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 2.92E+3nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 3.64E+3nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: 5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: 5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: 5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 6.18E+3nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 8.48E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University
Tohoku University
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair