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Found 80 with Last Name = 'tasaki' and Initial = 'm'
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517668(CHEMBL4578497)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097498(CHEMBL3586039)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517655(CHEMBL4547465)
Affinity DataIC50:  0.230nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097497(CHEMBL3586038)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517667(CHEMBL4540382)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517656(CHEMBL4580751)
Affinity DataIC50:  0.420nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517672(CHEMBL4575526)
Affinity DataIC50:  0.440nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517658(CHEMBL4524977)
Affinity DataIC50:  0.460nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097499(CHEMBL3586040)
Affinity DataIC50:  0.460nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517669(CHEMBL4594002)
Affinity DataIC50:  0.570nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517659(CHEMBL4439095)
Affinity DataIC50:  0.590nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517670(CHEMBL4529215)
Affinity DataIC50:  0.660nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097495(CHEMBL3586036)
Affinity DataIC50:  0.680nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517664(CHEMBL4526554)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517662(CHEMBL4466775)
Affinity DataIC50:  0.940nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517671(CHEMBL4545726)
Affinity DataIC50: <1nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517665(CHEMBL4455647)
Affinity DataIC50: <1nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469242(CHEMBL4283768)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517661(CHEMBL4464921)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097493(CHEMBL3586034)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469241(CHEMBL4289064)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517666(CHEMBL4585918)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517654(CHEMBL4441229)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097502(CHEMBL3586043)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469249(CHEMBL4294341)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097507(CHEMBL3586048)
Affinity DataIC50:  3nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517655(CHEMBL4547465)
Affinity DataIC50:  3nMAssay Description:Inhibition of PKCtheta in human Jurkat cells assessed as reduction in IL2 production after 14 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517658(CHEMBL4524977)
Affinity DataIC50: <3nMAssay Description:Inhibition of PKCtheta in human Jurkat cells assessed as reduction in IL2 production after 14 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469260(CHEMBL4281174)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469251(CHEMBL4287302)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097494(CHEMBL3586035)
Affinity DataIC50:  4nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469258(CHEMBL4294119)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097496(CHEMBL3586037)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469252(CHEMBL4287122)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469255(CHEMBL4286045)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469253(CHEMBL4279198)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469250(CHEMBL4281351)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of PKCtheta in human Jurkat cells transfected with pGL3-IL2 pro 43 plasmid assessed as suppression of IL-2 production after 14 hrs by fire...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469261(CHEMBL4290543)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50097503(CHEMBL3586044)
Affinity DataIC50:  10nMAssay Description:Inhibition of human full length PKCtheta assessed as fluorescence intensity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517672(CHEMBL4575526)
Affinity DataIC50:  10nMAssay Description:Inhibition of PKCtheta in human Jurkat cells assessed as reduction in IL2 production after 14 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517656(CHEMBL4580751)
Affinity DataIC50:  11nMAssay Description:Inhibition of PKCtheta in human Jurkat cells assessed as reduction in IL2 production after 14 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469262(CHEMBL4286223)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517662(CHEMBL4466775)
Affinity DataIC50:  16nMAssay Description:Inhibition of PKCtheta in human Jurkat cells assessed as reduction in IL2 production after 14 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCepsilon expressed in Baculovirus expression system using STK1-biotin as substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517669(CHEMBL4594002)
Affinity DataIC50:  17nMAssay Description:Inhibition of PKCtheta in human Jurkat cells assessed as reduction in IL2 production after 14 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517659(CHEMBL4439095)
Affinity DataIC50:  18nMAssay Description:Inhibition of PKCtheta in human Jurkat cells assessed as reduction in IL2 production after 14 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCdelta expressed in Baculovirus expression system using STK1-biotin as substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469242(CHEMBL4283768)
Affinity DataIC50:  22nMAssay Description:Inhibition of PKCtheta in human Jurkat cells transfected with pGL3-IL2 pro 43 plasmid assessed as suppression of IL-2 production after 14 hrs by fire...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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