Compile Data Set for Download or QSAR
maximum 50k data
Found 236 with Last Name = 'taylor' and Initial = 'sd'
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50108119(CHEMBL3600587)
Affinity DataKi:  1nMAssay Description:Reversible inhibition of STS (unknown origin) using 4-MUS as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50098106(CHEMBL24259 | PHENYLSULFAMATE | Sulfamic acid phen...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50098106(CHEMBL24259 | PHENYLSULFAMATE | Sulfamic acid phen...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50108118(CHEMBL3600594)
Affinity DataKi:  2.5nMAssay Description:Reversible inhibition of STS (unknown origin) using 4-MUS as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataKi:  10nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50363580(CHEMBL1945908)
Affinity DataKi:  23nMAssay Description:Inhibition of steroid sulfatase using 4-methylumbelliferyl sulfate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50243240((3-((R)-2-((S)-2-((S)-2-((S)-2-((S)-2-amino-3-carb...)
Affinity DataKi:  24nMAssay Description:Inhibition of human PTP1B expressed in Escherichia coli BL21(DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50243238(({2-Bromo-4-[40-bromo-30-(difluorosulfamoylmethyl)...)
Affinity DataKi:  24nMAssay Description:Inhibition of human PTP1B expressed in Escherichia coli BL21(DE3) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibition of cloned human transmembrane, tumor-associated isozyme CA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50051829(4-methyl-2-oxo-2H-chromen-7-yl sulfamate | CHEMBL1...)
Affinity DataKi:  25nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  30nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataKi:  30nMAssay Description:Inhibition of cloned human transmembrane, tumor-associated isozyme CA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175010((4-methyl-2-oxo-2H-chromen-7-yl)methanesulfonamide...)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataKi:  37nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  60nMAssay Description:Inhibition of recombinant human mitochondrial isozyme CA VAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50098106(CHEMBL24259 | PHENYLSULFAMATE | Sulfamic acid phen...)
Affinity DataKi:  63nMAssay Description:Inhibition of cloned human transmembrane, tumor-associated isozyme CA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370690(CHEMBL1628081)
Affinity DataKi:  80nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355360(CHEMBL1835425)
Affinity DataKi:  85nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 5 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  90nMAssay Description:Mixed type inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370691(CHEMBL1628004)
Affinity DataKi:  96nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175009((4-bromophenyl)difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  98nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175010((4-methyl-2-oxo-2H-chromen-7-yl)methanesulfonamide...)
Affinity DataKi:  98nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175002(CHEMBL198891 | difluoro(4-methyl-2-oxo-2H-chromen-...)
Affinity DataKi:  104nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50363580(CHEMBL1945908)
Affinity DataKi:  108nMAssay Description:Mixed type inhibition of steroid sulfatase using 4-methylumbelliferyl sulfate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175008((2-bromophenyl)difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  112nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175001(4-nitrophenyl-difluoromethanesulfonamide | CHEMBL3...)
Affinity DataKi:  113nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370690(CHEMBL1628081)
Affinity DataKi:  116nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175011(4-methylphenyl-difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  128nMAssay Description:Inhibition of recombinant human mitochondrial isozyme CA VAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370691(CHEMBL1628004)
Affinity DataKi:  129nMAssay Description:Inhibition of recombinant human mitochondrial isozyme CA VAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175001(4-nitrophenyl-difluoromethanesulfonamide | CHEMBL3...)
Affinity DataKi:  153nMAssay Description:Inhibition of recombinant human mitochondrial isozyme CA VAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175007(CHEMBL371870 | phenyldifluoromethanesulfonamide)
Affinity DataKi:  156nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175006(3-bromophenyl-difluoromethanesulfonamide | CHEMBL2...)
Affinity DataKi:  160nMAssay Description:Inhibition of recombinant human mitochondrial isozyme CA VAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175002(CHEMBL198891 | difluoro(4-methyl-2-oxo-2H-chromen-...)
Affinity DataKi:  195nMAssay Description:Inhibition of cloned human transmembrane, tumor-associated isozyme CA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370690(CHEMBL1628081)
Affinity DataKi:  208nMAssay Description:Inhibition of cloned human transmembrane, tumor-associated isozyme CA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175010((4-methyl-2-oxo-2H-chromen-7-yl)methanesulfonamide...)
Affinity DataKi:  240nMAssay Description:Inhibition of cloned human transmembrane, tumor-associated isozyme CA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  250nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175011(4-methylphenyl-difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  250nMAssay Description:Inhibition of cloned human transmembrane, tumor-associated isozyme CA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355372(CHEMBL482212)
Affinity DataKi:  250nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175009((4-bromophenyl)difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  273nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175011(4-methylphenyl-difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  348nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175007(CHEMBL371870 | phenyldifluoromethanesulfonamide)
Affinity DataKi:  357nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175002(CHEMBL198891 | difluoro(4-methyl-2-oxo-2H-chromen-...)
Affinity DataKi:  415nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175006(3-bromophenyl-difluoromethanesulfonamide | CHEMBL2...)
Affinity DataKi:  565nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175005(CHEMBL369953 | phenylmethanesulfonamide)
Affinity DataKi:  645nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370691(CHEMBL1628004)
Affinity DataKi:  670nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175008((2-bromophenyl)difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  714nMAssay Description:Inhibition of recombinant human mitochondrial isozyme CA VAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175007(CHEMBL371870 | phenyldifluoromethanesulfonamide)
Affinity DataKi:  785nMAssay Description:Inhibition of recombinant human mitochondrial isozyme CA VAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50107741(4-[3,5-di(4-difluorophosphonatephenethylcarboxamid...)
Affinity DataKi:  930nMAssay Description:Binding affinity towards the binding site in PTP1B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50175011(4-methylphenyl-difluoromethanesulfonamide | CHEMBL...)
Affinity DataKi:  952nMAssay Description:Inhibition of recombinant human cytosolic isozyme CA IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 236 total ) | Next | Last >>
Jump to: