Affinity DataKi: 730nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate assessed as unbound inhibitor concentration required for half maximal enz...More data for this Ligand-Target Pair
Affinity DataKi: 740nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate assessed as unbound inhibitor concentration required for half maximal ...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate assessed as residual enzyme activity after 2 to 10 mins by LC-MS/MS analy...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate assessed as residual enzyme activity after 2 to 10 mins by LC-MS/MS an...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 30 mins followed by 10-fold dilution and ...More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using testosterone as substrate preincubated for 30 mins followed by 10-fold dilution a...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using testosterone as substrate preincubated for 90 mins followed by 10-fold dilution a...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 90 mins followed by 10-fold dilution and ...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 30 mins followed by 10-fold dilution and ...More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using testosterone as substrate preincubated for 30 mins followed by 10-fold dilution a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 90 mins followed by 10-fold dilution and ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 90 mins followed by substrate addition by...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 30 mins followed by 10-fold dilution and ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 30 mins followed by 10-fold dilution and ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 90 mins followed by 10-fold dilution and ...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against HCV delta 21 NS5b RNA polymeraseMore data for this Ligand-Target Pair