BindingDB PrimarySearch_ki

Found 734 with Last Name = 'tran' and Initial = 'n'

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50328671((6aR,9R,10aR)-3-(1-hexylcyclobutyl)-6,6-dimethyl-6...)

Ki: 0.160nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603275(CHEMBL5187249)

Ki: 0.380nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603264(CHEMBL5206676)

Ki: 0.460nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603277(CHEMBL5194920)

Ki: 0.550nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603266(CHEMBL5203712)

Ki: 0.550nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Purchase PC cid PC sid

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603279(CHEMBL5203974)

Ki: 0.570nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603286(CHEMBL5183405)

Ki: 0.610nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603268(CHEMBL5206273)

Ki: 0.660nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603278(CHEMBL5176554)

Ki: 0.690nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557516(CHEMBL4787347)

Ki: 0.700nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50328664((6aR,10aR)-3-(1-Hexyl-cyclobut-1-yl)-6,6a,7,8,10,1...)

Ki: 0.840nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603288(CHEMBL5178005)

Ki: 0.920nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603284(CHEMBL5178943)

Ki: 1nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603281(CHEMBL5187812)

Ki: 1.10nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603283(CHEMBL5191435)

Ki: 1.10nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603274(CHEMBL5203428)

Ki: 1.20nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50328672((6aR,9R,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)

Ki: 1.40nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50328673((6aR,9S,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7...)

Ki: 1.5nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603280(CHEMBL5177375)

Ki: 1.5nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557512(CHEMBL4779775)

Ki: 1.60nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603285(CHEMBL5170526)

Ki: 1.90nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603272(CHEMBL5208446)

Ki: 1.90nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50557516(CHEMBL4787347)

Ki: 2nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557516(CHEMBL4787347)

Ki: 2.20nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50557513(CHEMBL4795739)

Ki: 2.30nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50328669((6aR,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6,6a,7,...)

Ki: 2.30nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Cannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557513(CHEMBL4795739)

Ki: 2.70nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557513(CHEMBL4795739)

Ki: 3.10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603265(CHEMBL5182571)

Ki: 3.40nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557514(CHEMBL4779296)

Ki: 3.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603271(CHEMBL5195537)

Ki: 4nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603276(CHEMBL5186742)

Ki: 4.60nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557517(CHEMBL4760082)

Ki: 4.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50557514(CHEMBL4779296)

Ki: 4.80nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603270(CHEMBL5209282)

Ki: 4.90nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557517(CHEMBL4760082)

Ki: 6.60nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603269(CHEMBL5176899)

Ki: 8.20nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603287(CHEMBL5169602)

Ki: 8.20nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50557517(CHEMBL4760082)

Ki: 8.40nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603273(CHEMBL5198520)

Ki: 8.80nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557514(CHEMBL4779296)

Ki: 9.5nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603267(CHEMBL5189278)

Ki: 11nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50557515(CHEMBL4744219)

Ki: 11nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50603263(CHEMBL5188390)

Ki: 18nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50557512(CHEMBL4779775)

Ki: 27nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL

PNG

BDBM50557511(CHEMBL4764017)

Ki: 29nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557512(CHEMBL4779775)

Ki: 32nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM50557515(CHEMBL4744219)

Ki: 35nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)

Ki: 36nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL DrugBank KEGG PC cid PC sid PDB Similars

Details Article PubMed DrugBank

Cannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL

PNG

BDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)

Ki: 40nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

CHEMBL DrugBank KEGG PC cid PC sid PDB Similars

Details Article PubMed

Displayed 1 to 50 (of 734 total ) | Next | Last >>

Filter my 734 hits

Targets 27▿
- Platelet-derived growth factor receptor beta 97
- Epidermal growth factor receptor 97
- Insulin-like growth factor 1 receptor 54
- Receptor tyrosine-protein kinase erbB-2 54
- Cannabinoid receptor 1 53
- Vascular endothelial growth factor receptor 1 52
- Beta-secretase 1 45
- Vascular endothelial growth factor receptor 2 43
- Fibroblast growth factor receptor 1 43
- Neutrophil elastase 34
- M-phase inducer phosphatase 2 30
- Probable periplasmic serine endoprotease DegP-like 29
- Dihydroorotate dehydrogenase (quinone), mitochondrial 22
- Proto-oncogene tyrosine-protein kinase Src 20
- Cannabinoid receptor 2 17
- Tyrosine-protein phosphatase non-receptor type 1 13
- Cruzipain 11
- Sialin 5
- Gag-Pol polyprotein [489-587] 3
- Dual specificity protein phosphatase 3 3
- Lipoprotein lipase 3
- Histone deacetylase 1
- Peroxisome proliferator-activated receptor gamma 1
- Bile acid receptor 1
- Retinoic acid receptor RXR-alpha 1
- Peroxisome proliferator-activated receptor alpha 1
- Vesicular acetylcholine transporter 1
- ...
Publications 17▿
- J Med Chem 41: 2588-603 (1998) 268
- J Med Chem 43: 2655-63 (2000) 100
- J Med Chem 42: 5120-30 (1999) 92
- Bioorg Med Chem Lett 22: 7345-50 (2012) 46
- Eur J Med Chem 230: (2022) 39
- Eur J Med Chem 230: (2022) 33
- Bioorg Med Chem Lett 38: (2021) 31
- Eur J Med Chem 224: (2021) 30
- J Med Chem 49: 4275-85 (2006) 28
- Eur J Med Chem 186: (2020) 22
- Bioorg Med Chem Lett 16: 1995-9 (2006) 17
- Eur J Med Chem 121: 387-398 (2016) 11
- Eur J Med Chem 103: 191-209 (2015) 7
- J Med Chem 63: 8231-8249 (2020) 5
- Bioorg Med Chem Lett 15: 135-8 (2004) 3
- Antimicrob Agents Chemother 52: 3467-77 (2008) 1
- Bioorg Med Chem 18: 6922-33 (2010) 1
Institutions 11▿
- Sugen 460
- University Of Otago 63
- University Of Paris 47
- National And Kapodistrian University Of Athens 39
- University Of Hawaii At Manoa 31
- Universite De La Mediterranee 28
- Universit£ 27
- University Of The Mediterranean 20
- Universidade Federal De Pernambuco 11
- Ume£ 7
- Walter Reed Army Institute Of Research 1
Affinity: 0.16 to 1.6E+5 nM▿
- Ki 59
- IC50 632
- EC50 43
- Affinity ≤ nM
Xtal structures: 4
Docked structures: 0
Catalog Cmpds: 41