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Found 38 with Last Name = 'tsoukala' and Initial = 'e'
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50316587(1-D-glucopyranosyl uracil | 1-beta-D-glucopyranosy...)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50316588(1-D-glucopyranosyl cytosine | 4-amino-1-beta-D-glu...)
Affinity DataKi:  7.70E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50240802(1-N-ACETYL-BETA-D-GLUCOSAMINE | CHEMBL335315 | N-(...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50316583(CHEMBL1095543 | N-(1-((2R,4S,6R)-4-fluoro-3,5-dihy...)
Affinity DataKi:  4.64E+4nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50316582(1-((2R,4S,6R)-4-fluoro-3,5-dihydroxy-6-(hydroxymet...)
Affinity DataKi:  3.46E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50316585(5-fluoro-1-((2R,4S,6R)-4-fluoro-3,5-dihydroxy-6-(h...)
Affinity DataKi:  3.67E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50316584(4-amino-1-((2R,4S,6R)-4-fluoro-3,5-dihydroxy-6-(hy...)
Affinity DataKi:  4.01E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50316586(CHEMBL1094537 | N-(1-((2R,4R,6R)-4-fluoro-5-hydrox...)
Affinity DataKi:  6.55E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50240803(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Affinity DataKi:  7.40E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340678(1-(beta-D-2-deoxy-erythro-pentofuranosyl)-5-fluoro...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340678(1-(beta-D-2-deoxy-erythro-pentofuranosyl)-5-fluoro...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 4 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340678(1-(beta-D-2-deoxy-erythro-pentofuranosyl)-5-fluoro...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340678(1-(beta-D-2-deoxy-erythro-pentofuranosyl)-5-fluoro...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340678(1-(beta-D-2-deoxy-erythro-pentofuranosyl)-5-fluoro...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 24...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340678(1-(beta-D-2-deoxy-erythro-pentofuranosyl)-5-fluoro...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340677((5-fluorouracil)5-Fluoro-1H-pyrimidine-2,4-dione |...)
Affinity DataIC50:  20nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340677((5-fluorouracil)5-Fluoro-1H-pyrimidine-2,4-dione |...)
Affinity DataIC50:  60nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 24...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340675((S)-5-fluoro-4-hydroxy-1-(3-oxo-3,6-dihydro-2H-pyr...)
Affinity DataIC50:  63nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340675((S)-5-fluoro-4-hydroxy-1-(3-oxo-3,6-dihydro-2H-pyr...)
Affinity DataIC50:  71nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 24...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340677((5-fluorouracil)5-Fluoro-1H-pyrimidine-2,4-dione |...)
Affinity DataIC50:  220nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 4 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340676(CHEMBL1762225 | exo-(S)-5-fluoro-4-hydroxy-1-(3-me...)
Affinity DataIC50:  430nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340679(CHEMBL1762230 | exo-1-((2S,4S,5R)-4,5-dihydroxy-3-...)
Affinity DataIC50:  570nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340677((5-fluorouracil)5-Fluoro-1H-pyrimidine-2,4-dione |...)
Affinity DataIC50:  600nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340675((S)-5-fluoro-4-hydroxy-1-(3-oxo-3,6-dihydro-2H-pyr...)
Affinity DataIC50:  830nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 4 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340675((S)-5-fluoro-4-hydroxy-1-(3-oxo-3,6-dihydro-2H-pyr...)
Affinity DataIC50:  950nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340676(CHEMBL1762225 | exo-(S)-5-fluoro-4-hydroxy-1-(3-me...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 24...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340679(CHEMBL1762230 | exo-1-((2S,4S,5R)-4,5-dihydroxy-3-...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 4 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340679(CHEMBL1762230 | exo-1-((2S,4S,5R)-4,5-dihydroxy-3-...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 24...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340679(CHEMBL1762230 | exo-1-((2S,4S,5R)-4,5-dihydroxy-3-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340677((5-fluorouracil)5-Fluoro-1H-pyrimidine-2,4-dione |...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340675((S)-5-fluoro-4-hydroxy-1-(3-oxo-3,6-dihydro-2H-pyr...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340679(CHEMBL1762230 | exo-1-((2S,4S,5R)-4,5-dihydroxy-3-...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340676(CHEMBL1762225 | exo-(S)-5-fluoro-4-hydroxy-1-(3-me...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 4 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340676(CHEMBL1762225 | exo-(S)-5-fluoro-4-hydroxy-1-(3-me...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340676(CHEMBL1762225 | exo-(S)-5-fluoro-4-hydroxy-1-(3-me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxyuridine after preincubation for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340676(CHEMBL1762225 | exo-(S)-5-fluoro-4-hydroxy-1-(3-me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50340675((S)-5-fluoro-4-hydroxy-1-(3-oxo-3,6-dihydro-2H-pyr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of thymidylate synthase in mouse L1210 cells assessed as inhibition of tritium release from [5-3H]deoxycytidine after preincubation for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed