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Found 38 with Last Name = 'tsuchida' and Initial = 'k'
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50539387(CHEMBL4648474)
Affinity DataIC50:  130nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50585028(CHEMBL5078185)
Affinity DataIC50:  190nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50525413(CHEMBL4448117)
Affinity DataIC50:  260nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50585029(CHEMBL5092917)
Affinity DataIC50:  300nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransforming growth factor beta-1 proprotein(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50585028(CHEMBL5078185)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of TGF beta 1 (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50525413(CHEMBL4448117)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180049(3-[2-isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180047(3-[2-isobutoxy-5-(3-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50539386(CHEMBL4646947)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransforming growth factor beta-1 proprotein(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50525413(CHEMBL4448117)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of TGF beta 1 (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151079((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180051((R)-4-(4-methylpentanoyl)-8-(4-methylpentylidene)-...)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180048((R)-8-(3-methylbutylidene)-4-(5-methylhexanoyl)-1-...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151090((S)-3-{(S)-2-[(S)-2-(2-Amino-acetylamino)-4-carbam...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151095((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151089((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151091((S)-3-{(S)-2-[(S)-2-(2-Amino-acetylamino)-4-carbam...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151088((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151087((S)-2-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151086((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151085((S)-3-[(S)-2-((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-4-c...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151084((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151083((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151081((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151080((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-((S)-2-Am...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151082((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-6-Amino-2-(...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151094((S)-3-{2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-acet...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151093((S)-4-(2-Amino-acetylamino)-4-{(S)-1-[(S)-2-carbox...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50151092((S)-3-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180050(3-[2-benzyloxy-5-(4-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  4.20E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180048((R)-8-(3-methylbutylidene)-4-(5-methylhexanoyl)-1-...)
Affinity DataIC50:  4.60E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180047(3-[2-isobutoxy-5-(3-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  6.00E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180049(3-[2-isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  6.10E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180051((R)-4-(4-methylpentanoyl)-8-(4-methylpentylidene)-...)
Affinity DataIC50:  6.50E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180052(3-[5-(4-isobutoxybenzoyl)-2-propoxyphenyl]propioni...)
Affinity DataIC50:  9.10E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180046(3-[2-isobutoxy-5-(4-propoxybenzoyl)phenyl]propioni...)
Affinity DataIC50:  9.30E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180053(3-(5-benzoyl-2-isobutoxyphenyl)propionic acid | CH...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180045(3-[3-(4-isobutoxybenzoyl)phenyl]propionic acid | C...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed