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Found 104 with Last Name = 'tsujita' and Initial = 'r'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.440nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290098((R)-3-Cyclohexylmethyl-1,8,8-trimethyl-3-aza-bicyc...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290099((S)-3-(4-Cyclohexyl-butyl)-1,8,8-trimethyl-3-aza-b...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290100((S)-3-Cyclohexylmethyl-1,8,8-trimethyl-3-aza-bicyc...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290095((R)-3-(2-Cyclohexyl-ethyl)-1,8,8-trimethyl-3-aza-b...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290096((S)-3-(2-Cyclopentyl-ethyl)-1,8,8-trimethyl-3-aza-...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290094((S)-3-(2-Cyclohexyl-ethyl)-1,8,8-trimethyl-3-aza-b...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290101((S)-3-(3-Cyclohexyl-propyl)-1,8,8-trimethyl-3-aza-...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290093((S)-3-(2-Cyclooctyl-ethyl)-1,8,8-trimethyl-3-aza-b...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290092((S)-3-(2-Cycloheptyl-ethyl)-1,8,8-trimethyl-3-aza-...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290097((S)-3-Cyclohexyl-1,8,8-trimethyl-3-aza-bicyclo[3.2...)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290091((S)-3-(2-Adamantan-2-yl-ethyl)-1,8,8-trimethyl-3-a...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM81982(CAS_97-39-2 | DITOLYLGUANIDINE | DTG | Di-o-tolylg...)
Affinity DataKi:  27nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50001044((1S,9S,13S)-10-allyl-1,13-dimethyl-10-azatricyclo[...)
Affinity DataKi:  157nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151161(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  220nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151159(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  280nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151163(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  870nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151168(5-Phenyl-1H-pyrrole-2-carboxylic acid (cyclohexylc...)
Affinity DataKi:  910nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151160(5-Phenyl-1H-pyrrole-2-carboxylic acid (3-diethylam...)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151169(5-Phenyl-1H-pyrrole-2-carboxylic acid [1-cyclohexy...)
Affinity DataKi:  1.17E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151158(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-tert-buty...)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151167(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  1.29E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151164(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  1.32E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151157(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  1.37E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151165(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  1.92E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151170(CHEMBL185887 | N-[Cyclohexylcarbamoyl-(4-fluoro-ph...)
Affinity DataKi:  2.03E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151166(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  2.63E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151162((S)-3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346122(2-(4-(2-(4-bromo-5-methylthiophen-2-yl)-5-ethyl-6-...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346123(2-(4-(5-ethyl-2-(5-fluorothiophen-2-yl)-6-methylpy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346121(2-(4-(2-(5-chlorothiophen-2-yl)-5-ethyl-6-methylpy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346120(2-(4-(2-(5-bromothiophen-2-yl)-5-ethyl-6-methylpyr...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human PDE4D3 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346100(4-(5-allyl-6-ethyl-2-phenylpyrimidin-4-ylamino)ben...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346119(2-(4-(5-ethyl-6-methyl-2-(5-(methylthio)thiophen-2...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346104(4-(5-allyl-6-methyl-2-(thiophen-3-yl)pyrimidin-4-y...)
Affinity DataIC50:  68nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346112(4-(5-allyl-2-(5-methoxythiophen-2-yl)-6-methylpyri...)
Affinity DataIC50:  78nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346100(4-(5-allyl-6-ethyl-2-phenylpyrimidin-4-ylamino)ben...)
Affinity DataIC50:  82nMAssay Description:Inhibition of human PDE4D3 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346103(4-(5-allyl-6-methyl-2-(thiophen-2-yl)pyrimidin-4-y...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346096(4-(5-cyano-6-methyl-2-phenylpyrimidin-4-ylamino)be...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346091(4-(5-ethyl-6-methyl-2-phenylpyrimidin-4-ylamino)be...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346111(4-(5-allyl-6-methyl-2-(5-methylthiophen-2-yl)pyrim...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346089(4-(5-allyl-6-methyl-2-phenylpyrimidin-4-ylamino)be...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346118(2-(4-(5-allyl-2-(5-methoxythiophen-2-yl)-6-methylp...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346109(4-(5-allyl-6-methyl-2-m-tolylpyrimidin-4-ylamino)b...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346108(4-(5-allyl-6-methyl-2-p-tolylpyrimidin-4-ylamino)b...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346110(4-(5-allyl-2-(4-methoxyphenyl)-6-methylpyrimidin-4...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346098(4-(5-formyl-6-methyl-2-phenylpyrimidin-4-ylamino)b...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50346117(2-(4-(5-allyl-6-methyl-2-(5-methylthiophen-2-yl)py...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human PDE4B1 incubated for 10 mins using cAMP and [3H]cAMP substratesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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