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Found 194 with Last Name = 'ullrich' and Initial = 'jw'
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  10nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(CHEMBL153469 | N-Hydroxy-3-(4-methoxy-benzenesulfo...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  30nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  50nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  50nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  60nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  200nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(CHEMBL153469 | N-Hydroxy-3-(4-methoxy-benzenesulfo...)
Affinity DataKi:  300nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  500nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  600nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  600nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  700nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(CHEMBL153469 | N-Hydroxy-3-(4-methoxy-benzenesulfo...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.100nMAssay Description:Progesterone receptor antagonist activity based on its ability to block progesterone induced alkaline phosphatase in the human breast cancer cell lin...More data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305075(3-benzyl-4-(3-(3-(methylsulfonyl)phenoxy)phenyl)-8...)
Affinity DataIC50:  0.920nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305077(3-methyl-4-(3-(3-(methylsulfonyl)phenoxy)phenyl)-8...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305072(8-chloro-3-methyl-4-(3-(3-(methylsulfonyl)phenoxy)...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305073(3-benzyl-8-chloro-4-(3-(3-(methylsulfonyl)phenoxy)...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305064(3-(3-(3-(3-methyl-8-(trifluoromethyl)quinolin-4-yl...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50317735(3-benzyl-4-(3'-(methylsulfonyl)biphenyl-3-yl)-8-(t...)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [3H]T0901317 from LXRbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305070(4-(3-(3-(ethylsulfonyl)phenoxy)phenyl)-3-methyl-8-...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50317744(4-(4'-fluoro-3'-(methylsulfonyl)biphenyl-3-yl)-3-m...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [3H]T0901317 from LXRbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305068(4-(3-(3-(isopropylsulfonyl)phenoxy)phenyl)-3-methy...)
Affinity DataIC50:  1.80nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50317733(3-methyl-4-(3'-(methylsulfonyl)biphenyl-3-yl)-8-(t...)
Affinity DataIC50:  1.80nMAssay Description:Displacement of [3H]T0901317 from LXRbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305060(4-(3-(3-fluoro-5-(methylsulfonyl)phenoxy)phenyl)-3...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305075(3-benzyl-4-(3-(3-(methylsulfonyl)phenoxy)phenyl)-8...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRbeta-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305077(3-methyl-4-(3-(3-(methylsulfonyl)phenoxy)phenyl)-8...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRbeta-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50317737(3-ethyl-4-(3'-(methylsulfonyl)biphenyl-3-yl)-8-(tr...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [3H]T0901317 from LXRbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305067(4-(3-(3-(isopropylsulfonyl)phenoxy)phenyl)-8-(trif...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305069(3-methyl-4-(3-(3-(propylsulfonyl)phenoxy)phenyl)-8...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50317746(4-(4'-fluoro-3'-(methylsulfonyl)biphenyl-3-yl)-8-(...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H]T0901317 from LXRbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305074(4-(3-(3-(methylsulfonyl)phenoxy)phenyl)-8-(trifluo...)
Affinity DataIC50:  2.80nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM35094(biarylether alcohol quinoline, 5f)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305059(4-(3-(3-chloro-5-(methylsulfonyl)phenoxy)phenyl)-3...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human LBD of ERbetaMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305062(4-(3-(3-(3-methoxypropylsulfonyl)phenoxy)phenyl)-3...)
Affinity DataIC50:  3.20nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRalpha-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50317742(3-methyl-4-(4'-methyl-3'-(methylsulfonyl)biphenyl-...)
Affinity DataIC50:  3.20nMAssay Description:Displacement of [3H]T0901317 from LXRbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50317745(4-(2',4'-difluoro-5'-(methylsulfonyl)biphenyl-3-yl...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [3H]T0901317 from LXRbeta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50305073(3-benzyl-8-chloro-4-(3-(3-(methylsulfonyl)phenoxy)...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [3H]T0901317 from human recombinant LXRbeta-LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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