Affinity DataKi: 0.150nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]DPCPX (without GTP) from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [3H]DPCPX (with GTP) from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]-8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition si...More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:In vitro displacement of [3H]-spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Binding affinity for adenosine A1 receptor from rat cortical membrane using [3H]DPCPX without GTPMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center For Drug Research
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Displacement of [3H]DPCPX (without GTP) from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair