Compile Data Set for Download or QSAR
maximum 50k data
Found 298 with Last Name = 'walker' and Initial = 'b'
TargetProcathepsin L(Homo sapiens (Human))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090644(CHEMBL48837 | {(S)-1-[(S)-1-(4-Butoxy-benzyl)-2,3-...)
Affinity DataKi:  0.600nMAssay Description:Ability to block cathepsin L-catalyzed hydrolysis of the fluorogenic substrate Z-Phe-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090645((S)-2-Benzyl-N-[(S)-4-guanidino-1-(2-oxo-acetyl)-b...)
Affinity DataKi:  40nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
The Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50089610((Z)-(S)-5-Amino-7-methyl-4-oxo-oct-2-enoic acid me...)
Affinity DataKi:  76nMAssay Description:Inhibitory activity of the compound against leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090645((S)-2-Benzyl-N-[(S)-4-guanidino-1-(2-oxo-acetyl)-b...)
Affinity DataKi:  90nMAssay Description:Ability to block cathepsin L-catalyzed hydrolysis of the fluorogenic substrate Z-Phe-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Queen'S University of Belfast

LigandPNGBDBM81670(Peptidyl ene diones, COOEt)
Affinity DataKi:  94nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Queen'S University of Belfast

LigandPNGBDBM81671(Peptidyl ene diones, COOMe)
Affinity DataKi:  125nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090644(CHEMBL48837 | {(S)-1-[(S)-1-(4-Butoxy-benzyl)-2,3-...)
Affinity DataKi:  214nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090646((S)-2-Acetylamino-5-guanidino-pentanoic acid [(S)-...)
Affinity DataKi:  640nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311228((S)-2-((S)-3-(4-hydroxyphenyl)-2-(2-mercaptoacetam...)
Affinity DataKi:  770nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Queen'S University of Belfast

LigandPNGBDBM81670(Peptidyl ene diones, COOEt)
Affinity DataKi:  850nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090643((S)-2-Acetylamino-4-methyl-pentanoic acid {(S)-1-[...)
Affinity DataKi:  970nMAssay Description:Ability to block cathepsin L-catalyzed hydrolysis of the fluorogenic substrate Z-Phe-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311181((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-3-(1...)
Affinity DataKi:  1.10E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090643((S)-2-Acetylamino-4-methyl-pentanoic acid {(S)-1-[...)
Affinity DataKi:  1.25E+3nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311166((2S,3R)-N-((S)-1-amino-4-methyl-1-oxopentan-2-yl)-...)
Affinity DataKi:  1.30E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311165((2S,3R)-N-((S)-1-amino-3-methyl-1-oxobutan-2-yl)-2...)
Affinity DataKi:  1.80E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311225((S)-5-guanidino-2-((S)-3-(4-hydroxyphenyl)-2-(2-me...)
Affinity DataKi:  3.00E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311184((S)-2-((S)-3-(1H-indol-3-yl)-2-(2-mercaptoacetamid...)
Affinity DataKi:  3.70E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311193((S)-6-amino-2-((S)-2-(2-mercaptoacetamido)-4-(meth...)
Affinity DataKi:  3.90E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311183((S)-2-((S)-3-(1H-indol-3-yl)-2-(2-mercaptoacetamid...)
Affinity DataKi:  4.10E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311230((S)-4-amino-3-((S)-3-(4-hydroxyphenyl)-2-(2-mercap...)
Affinity DataKi:  5.50E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311226((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-3-(4...)
Affinity DataKi:  6.50E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311194((S)-5-guanidino-2-((S)-2-(2-mercaptoacetamido)-4-(...)
Affinity DataKi:  6.60E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311198((S)-4-amino-3-((S)-2-(2-mercaptoacetamido)-4-(meth...)
Affinity DataKi:  7.00E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311148((S)-6-amino-2-((S)-3-(4-hydroxyphenyl)-2-(2-mercap...)
Affinity DataKi:  8.50E+3nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311217((S)-N-((S)-1-amino-3-methyl-1-oxobutan-2-yl)-2-(2-...)
Affinity DataKi:  1.00E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311179((S)-2-((S)-3-(1H-indol-3-yl)-2-(2-mercaptoacetamid...)
Affinity DataKi:  1.00E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311171((S)-2-((S)-2-(2-mercaptoacetamido)-3-phenylpropana...)
Affinity DataKi:  1.10E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311173((S)-6-amino-2-((S)-2-(2-mercaptoacetamido)-4-methy...)
Affinity DataKi:  1.40E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311227((S)-N-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2...)
Affinity DataKi:  1.40E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291657(4-Methoxy-benzoic acid 2-{[1-(2-tert-butoxycarbony...)
Affinity DataKi:  1.40E+4nMAssay Description:Evaluated for inhibition against thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311151((S)-N-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2...)
Affinity DataKi:  1.80E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311191((S)-2-((S)-2-(2-mercaptoacetamido)propanamido)-4-m...)
Affinity DataKi:  2.10E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311150((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-3-(1...)
Affinity DataKi:  2.10E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311214((S)-6-amino-2-((S)-2-(2-mercaptoacetamido)-3-methy...)
Affinity DataKi:  2.20E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311180((S)-2-((S)-3-(1H-indol-3-yl)-2-(2-mercaptoacetamid...)
Affinity DataKi:  2.50E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311231((S)-2-((S)-3-(4-hydroxyphenyl)-2-(2-mercaptoacetam...)
Affinity DataKi:  2.70E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311229((S)-2-((S)-3-(4-hydroxyphenyl)-2-(2-mercaptoacetam...)
Affinity DataKi:  3.30E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311210((S)-N1-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(...)
Affinity DataKi:  3.70E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311185((S)-3-((S)-3-(1H-indol-3-yl)-2-(2-mercaptoacetamid...)
Affinity DataKi:  3.80E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311152((S)-2-((S)-3-(1H-imidazol-4-yl)-2-(2-mercaptoaceta...)
Affinity DataKi:  4.70E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311182((S)-N-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2...)
Affinity DataKi:  4.90E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311221((S)-2-(2-(2-mercaptoacetamido)acetamido)-3-phenylp...)
Affinity DataKi:  5.10E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311190((S)-2-((S)-2-(2-mercaptoacetamido)propanamido)-3-m...)
Affinity DataKi:  5.10E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311177((S)-N-((S)-1-amino-4-methyl-1-oxopentan-2-yl)-2-(2...)
Affinity DataKi:  5.30E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311200((S)-N-((S)-1-amino-5-guanidino-1-oxopentan-2-yl)-1...)
Affinity DataKi:  5.60E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311242((2S,3R)-N-((S)-1-amino-3-(1H-indol-3-yl)-1-oxoprop...)
Affinity DataKi:  6.50E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311215((S)-5-guanidino-2-((S)-2-(2-mercaptoacetamido)-3-m...)
Affinity DataKi:  6.90E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311218((S)-2-((S)-2-(2-mercaptoacetamido)-3-methylbutanam...)
Affinity DataKi:  6.90E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311211((S)-N1-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-...)
Affinity DataKi:  7.00E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50311216((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...)
Affinity DataKi:  7.20E+4nMpH: 7.2Assay Description:Inhibition of Pseudomonas aeruginosa LasB by fluorimetric assay in buffer of pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 298 total ) | Next | Last >>
Jump to: