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Found 703 with Last Name = 'wang' and Initial = 'yl'
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataKi:  190nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518879(CHEMBL4450911)
Affinity DataKi:  2.03E+3nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518902(CHEMBL4458011)
Affinity DataKi:  2.41E+3nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518878(CHEMBL4464588)
Affinity DataKi:  3.36E+3nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518889(CHEMBL4560468)
Affinity DataKi:  4.16E+3nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518901(CHEMBL4468952)
Affinity DataKi:  6.37E+3nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518882(CHEMBL4471138)
Affinity DataKi:  6.84E+3nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518890(CHEMBL4439726)
Affinity DataKi:  1.08E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518907(CHEMBL4472399)
Affinity DataKi:  1.35E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518892(CHEMBL4453017)
Affinity DataKi:  1.42E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518895(CHEMBL4454286)
Affinity DataKi:  1.54E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518887(CHEMBL4527309)
Affinity DataKi:  1.58E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518906(CHEMBL4444728)
Affinity DataKi:  1.87E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518899(CHEMBL4460555)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518891(CHEMBL4460127)
Affinity DataKi:  3.27E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518886(CHEMBL4471673)
Affinity DataKi:  3.28E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518881(CHEMBL4455145)
Affinity DataKi:  3.57E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518884(CHEMBL4588584)
Affinity DataKi:  3.63E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518897(CHEMBL4450628)
Affinity DataKi:  4.10E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518893(CHEMBL4545947)
Affinity DataKi:  6.79E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518896(CHEMBL4517893)
Affinity DataKi:  6.86E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518877(CHEMBL4546207)
Affinity DataKi:  7.06E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518908(CHEMBL4543432)
Affinity DataKi:  8.07E+4nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518883(CHEMBL4577981)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518885(CHEMBL4451026)
Affinity DataKi:  1.14E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518903(CHEMBL4445648)
Affinity DataKi:  1.66E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518905(CHEMBL4469059)
Affinity DataKi:  1.71E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518900(CHEMBL4545274)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518894(CHEMBL4444926)
Affinity DataKi:  2.16E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518898(CHEMBL4546893)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518904(CHEMBL4544829)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518880(CHEMBL4438924)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518909(CHEMBL4464521)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50518888(CHEMBL4466256)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of bacterial N-terminal His-tagged TEV protease site linked TEM-1 (24 to 286 amino acids) expressed in Escherichia coli Transetta (DE3) pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50:  0.400nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in rat C6 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated f...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50351665(CHEMBL1822369)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50351664(CHEMBL1822368)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50351662(CHEMBL1822366)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50351633(CHEMBL497118)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50351579(CHEMBL494985)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM24460(N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM28028(2-aminopyridine analogue, 7 | N-{4-[(2-amino-3-eth...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50351641(CHEMBL1823128)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM28030(2-aminopyridine analogue, 9 | N-{4-[(2-amino-3-chl...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM24462(N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM24459(N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50351650(CHEMBL1823252)
Affinity DataIC50:  1nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM24463(N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM24457(2-[(3-fluoro-4-{1H-pyrrolo[2,3-b]pyridin-4-yloxy}p...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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