Affinity DataKi: 0nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of L-1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of L-1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.00200nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of L-1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >0.00400nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of L-1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >0.00400nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of L-1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >0.00400nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of L-1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >0.00400nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of L-1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0871nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of horse liver alcohol dehydrogenase enzyme by Non-competitive inhibitionMore data for this Ligand-Target Pair
TargetAlcohol dehydrogenase 1A(Homo sapiens (Human))
University Of Rochester Medical Center
Curated by ChEMBL
University Of Rochester Medical Center
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Apparent inhibition constant against mammalian liver alcohol dehydrogenase (ADH)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor delta 1 using [3H]DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
TargetAlcohol dehydrogenase 1A(Homo sapiens (Human))
University Of Rochester Medical Center
Curated by ChEMBL
University Of Rochester Medical Center
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition constant against mammalian liver alcohol dehydrogenase (ADH)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II isoform); Range is 6-10 nMMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I isoform); Range is 33-37 nMMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor delta 1 using [3H]DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Chiba University
Curated by ChEMBL
Chiba University
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor kappa 1 using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Chiba University
Curated by ChEMBL
Chiba University
Curated by ChEMBL
Affinity DataKi: 123nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor kappa 1 using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor delta 1 using [3H]DPDPE as radioligandMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II isoform)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetAlcohol dehydrogenase 1A(Homo sapiens (Human))
University Of Rochester Medical Center
Curated by ChEMBL
University Of Rochester Medical Center
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition constant against mammalian liver alcohol dehydrogenase (ADH)More data for this Ligand-Target Pair
Affinity DataKi: 417nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor delta 1 using [3H]DPDPE as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Chiba University
Curated by ChEMBL
Chiba University
Curated by ChEMBL
Affinity DataKi: 468nMAssay Description:Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor kappa 1 using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 2 (IMPDH type II)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 1(Homo sapiens (Human))
Codon Pharmaceuticals
Curated by ChEMBL
Codon Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 890nMAssay Description:Inhibitory activity against human Inosine-5'-monophosphate dehydrogenase 1 (IMPDH type I)More data for this Ligand-Target Pair