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Found 141 with Last Name = 'wells' and Initial = 'e'
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336715(4-(3,3-Dimethyl-butyrylamino)-3,5-difluoro-N-thiaz...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336712(4-(3,3-Dimethyl-butyrylamino)-3-fluoro-N-thiazol-2...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336719(4-(3,3-Dimethyl-butyrylamino)-5-fluoro-2-methoxy-N...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336717(4-(3,3-Dimethyl-butyrylamino)-3-methoxy-N-thiazol-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336714(4-(3,3-Dimethyl-butyrylamino)-3-methyl-N-thiazol-2...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336723(3-Chloro-4-(3,3-dimethyl-butyrylamino)-N-thiazol-2...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336720(CHEMBL1671923 | N-(5-Chloro-thiazol-2-yl)-4-(3,3-d...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336713(3-Chloro-4-(3,3-dimethyl-butyrylamino)-5-methyl-N-...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336729(4-(3,3-Dimethyl-butyrylamino)-N-thiazol-2-yl-benza...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336709(4-(3,3-Dimethyl-butyrylamino)-2-methoxy-N-thiazol-...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336728(4-(3-Methyl-butyrylamino)-N-thiazol-2-yl-benzamide...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336727(CHEMBL1671928 | N-(2,2-Dimethyl-propyl)-N'-thiazol...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336710(4-(3,3-Dimethyl-butyrylamino)-N-(5-methyl-thiazol-...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336726(2-Chloro-4-(3,3-dimethyl-butyrylamino)-N-thiazol-2...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336725(4-pentanamido-N-(thiazol-2-yl)benzamide | CHEMBL16...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336724(4-(3,3-Dimethyl-butyrylamino)-2-methyl-N-thiazol-2...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336723(3-Chloro-4-(3,3-dimethyl-butyrylamino)-N-thiazol-2...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336722(2-methyl-N-(4-(thiazol-2-ylcarbamoyl)phenyl)benzam...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336721(4-(3,3-Dimethyl-butyrylamino)-N-(4,5-dimethyl-thia...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336719(4-(3,3-Dimethyl-butyrylamino)-5-fluoro-2-methoxy-N...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336720(CHEMBL1671923 | N-(5-Chloro-thiazol-2-yl)-4-(3,3-d...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336715(4-(3,3-Dimethyl-butyrylamino)-3,5-difluoro-N-thiaz...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]-MRS1754 from human recombinant adenosine A2B receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336718(4-Isobutyrylamino-N-thiazol-2-yl-benzamide | CHEMB...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336717(4-(3,3-Dimethyl-butyrylamino)-3-methoxy-N-thiazol-...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336716(4-Butyrylamino-N-thiazol-2-yl-benzamide | CHEMBL16...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336715(4-(3,3-Dimethyl-butyrylamino)-3,5-difluoro-N-thiaz...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336714(4-(3,3-Dimethyl-butyrylamino)-3-methyl-N-thiazol-2...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336713(3-Chloro-4-(3,3-dimethyl-butyrylamino)-5-methyl-N-...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336712(4-(3,3-Dimethyl-butyrylamino)-3-fluoro-N-thiazol-2...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336711(4-Propionylamino-N-thiazol-2-yl-benzamide | CHEMBL...)
Affinity DataKi:  890nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336710(4-(3,3-Dimethyl-butyrylamino)-N-(5-methyl-thiazol-...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336709(4-(3,3-Dimethyl-butyrylamino)-2-methoxy-N-thiazol-...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50336715(4-(3,3-Dimethyl-butyrylamino)-3,5-difluoro-N-thiaz...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO-K1 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110881(4-(2-oxo-3-(4-(5-phenylpentylthio)phenoxy)propoxy)...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by bilayer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110846(4-(3-(4-(decyloxy)phenoxy)-2-oxopropoxy)benzoic ac...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by bilayer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110859(CHEMBL26200 | {4-[3-(4-Decyloxy-phenoxy)-2-oxo-pro...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110854(4-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxy]-3-nitro-b...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110873(4-[3-(4-Dodecyloxy-phenoxy)-2-oxo-propoxy]-benzoic...)
Affinity DataIC50:  26nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110875(5-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxy]-pentanoic...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110846(4-(3-(4-(decyloxy)phenoxy)-2-oxopropoxy)benzoic ac...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110865(3-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxymethyl]-ben...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110872(4-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxymethyl]-ben...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110884(4-[3-(4-Octyloxy-phenoxy)-2-oxo-propoxy]-benzoic a...)
Affinity DataIC50:  46nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110879(4-{2-Oxo-3-[4-(5-phenyl-pentyloxy)-phenoxy]-propox...)
Affinity DataIC50:  48nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110888(3-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxy]-benzoic a...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110860(CHEMBL29247 | {3-[3-(4-Decyloxy-phenoxy)-2-oxo-pro...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by soluble assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2 beta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50110853(CHEMBL29246 | {3-[3-(4-Decyloxy-phenoxy)-2-oxo-pro...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against cytosolic Phospholipase A2 (PLA2) by bilayer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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