TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of human HGPRT using fixed concentration of guanine and variable concentrations of PRib-PP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of recombinant human HGPRT using fixed concentration of guanine and variable concentrations of PRib-PP as substrate by Hanes plot analysisMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of recombinant human HGPRT using fixed concentration of guanine and variable concentrations of PRib-PP as substrate by Hanes plot analysisMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of human HGPRT using fixed concentration of guanine and variable concentrations of PRib-PP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibitory activity against rabbit muscle glycogen phosphorylase a in the absence of AMPMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of human HGPRT using fixed concentration of guanine and variable concentrations of PRib-PP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant N-terminal 6His-tagged HGPRT expressed in Escherichia coli BL21 (DE3) using fixed concentration ...More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant N-terminal 6His-tagged HGPRT expressed in Escherichia coli BL21 (DE3) using fixed concentration ...More data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant N-terminal 6His-tagged HGPRT expressed in Escherichia coli BL21 (DE3) using fixed concentration ...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant N-terminal 6His-tagged HGPRT expressed in Escherichia coli BL21 (DE3) using fixed concentration ...More data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant N-terminal 6His-tagged HGPRT expressed in Escherichia coli BL21 (DE3) using fixed concentration ...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Inhibitory activity against pig Liver glycogen phosphorylase aMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant N-terminal 6His-tagged HGPRT expressed in Escherichia coli BL21 (DE3) using fixed concentration ...More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of human HGPRT using fixed concentration of guanine and variable concentrations of PRib-PP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 630nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 640nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 640nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetHypoxanthine-guanine phosphoribosyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant N-terminal 6His-tagged HGPRT expressed in Escherichia coli BL21 (DE3) using fixed concentration ...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 750nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 790nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 960nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of St. Andrews
Curated by ChEMBL
University Of St. Andrews
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair