Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]SCH58261 from human recombinant A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]SCH58261 from human recombinant A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Antagonist activity at rat A2A receptor by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity towards human melanocortin 4 receptor expressed in HEK 293 cells using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity to C57BL/6J mouse MC4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity towards human melanocortin 4 receptor expressed in HEK 293 cells using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Antagonist activity at rat A2A receptor by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity towards human melanocortin 4 receptor expressed in HEK 293 cells using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]SCH58261 from human recombinant A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Binding affinity to rat MC4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Displacement of [3H]SCH58261 from human recombinant A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards human melanocortin 4 receptor expressed in HEK 293 cells using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Tested for inhibitory activity against calpain.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]SCH58261 from human recombinant A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity towards human melanocortin 4 receptor expressed in HEK 293 cells using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonist activity at rat A2A receptor by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]SCH58261 from human recombinant A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]SCH58261 from human recombinant A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Activity at MC4R assessed as inhibition of alpha-MSH-stimulated cAMP productionMore data for this Ligand-Target Pair