TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Steady state and transient kinetics to a freely reversible, non-covalently bound, human recombinant Phospholipase A2 (rhLp-PLA2) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]PGD2 from CRTH2 expressed in HEK293 cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 expressed in K562 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonistic activity at CRTH2 in human eosinophils assessed as inhibition of PGD2-induced calcium mobilization after 60 mins by Fluo-3 based fluores...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]PGD2 from CRTH2 expressed in CHO cells after 1 hr by beta counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Antagonistic activity at CRTH2 in human eosinophils assessed as inhibition of PGD2-induced calcium mobilization after 60 mins by Fluo-3 based fluores...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonistic activity at CRTH2 in human eosinophils assessed as inhibition of PGD2-induced calcium mobilization after 60 mins by Fluo-3 based fluores...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Antagonistic activity at CRTH2 in human eosinophils assessed as inhibition of PGD2-induced calcium mobilization after 60 mins by Fluo-3 based fluores...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals
Curated by ChEMBL
British Biotech Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Compound was evaluated for inhibition of peptide deformylase, PDF.Fe of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 expressed in K562 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Antagonistic activity at CRTH2 in human eosinophils assessed as inhibition of PGD2-induced calcium mobilization after 60 mins by Fluo-3 based fluores...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:In vitro binding affinity (agonistic) towards human CRTH2 receptor expressed in CHO cells; range 15 to 25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Antagonistic activity at CRTH2 in human eosinophils assessed as inhibition of PGD2-induced calcium mobilization after 60 mins by Fluo-3 based fluores...More data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 143nMAssay Description:Displacement of [3H]PGD2 from CRTH2 expressed in CHO cells after 1 hr by beta counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 225nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 299nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 457nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 634nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 979nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 1.87E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals
Curated by ChEMBL
British Biotech Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Compound was evaluated for inhibition of peptide deformylase, PDF.Ni of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 2.98E+3nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.86E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.89E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.71E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cells; range 25 nM to 8 uMMore data for this Ligand-Target Pair
Affinity DataKi: 8.46E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair