TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:In vitro binding affinity on cloned Serotonin transporterMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:In vitro binding affinity on cloned Serotonin transporterMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity on cloned Serotonin transporterMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 1.89nMAssay Description:In vitro binding affinity on cloned Serotonin transporterMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
Affinity DataKi: 38nMAssay Description:Inhibition of human GSK-3beta using biotin-AAEELDSRAGS(PO3H2)PQL as substrate after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
Affinity DataKi: 77nMAssay Description:Displacement of [3H]-CGP12177 from beta1-adrenergic receptor in rat heart membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 115nMAssay Description:In vitro binding affinity on cloned Dopamine transporterMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
Affinity DataKi: 770nMAssay Description:Inhibition of GSK-3beta using phospho-glycogen synthase peptide-2 as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 1.21E+3nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 1.35E+3nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 1.42E+3nMAssay Description:In vitro binding affinity on cloned Dopamine transporterMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:In vitro binding affinity on cloned Norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 2.04E+3nMAssay Description:In vitro binding affinity on cloned Dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of [125I]-Iodopindolol from beta1-adrenergic receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [125I]-Iodopindolol from beta1-adrenergic receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataKi: 2.65E+3nMAssay Description:In vitro binding affinity on cloned Dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [125I]-Iodopindolol from beta1-adrenergic receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
Affinity DataKi: 7.70E+3nMAssay Description:Displacement of [125I]-Iodopindolol from beta2-adrenergic receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Iodopindolol from beta2-adrenergic receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Iodopindolol from beta2-adrenergic receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 90 mins prior to ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 0.813nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate preincubated for 60 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair