Compile Data Set for Download or QSAR
maximum 50k data
Found 2081 with Last Name = 'wood' and Initial = 'l'
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM412656(US10399974, Example 54)
Affinity DataKi:  0.0470nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM241208(US11046688, Example 50 | US9409907, 50)
Affinity DataKi:  0.0840nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50464039(CHEMBL4245639)
Affinity DataKi:  0.0880nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM241333(US10479788, Example 177 | US11046688, Example 177 ...)
Affinity DataKi:  0.0940nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM412611(N-(2-ethoxy-4-(4-methyl-4H-1,2,4-triazol-3-yl)phen...)
Affinity DataKi:  0.110nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM241338(US10479788, Example 182 | US11046688, Example 182 ...)
Affinity DataKi:  0.110nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50464037(CHEMBL4240502)
Affinity DataKi:  0.120nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM412614(N2-(4-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)-2-ethox...)
Affinity DataKi:  0.120nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM241335(US9409907, 179)
Affinity DataKi:  0.130nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50464040(CHEMBL4251352)
Affinity DataKi:  0.190nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM241235(US10479788, Example 77 | US11046688, Example 77 | ...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of human full length MPS1 expressed in recombinant baculovirus infected Sf9 insect cells using 5FAM-DHTGFLTEYVATRCONH2 as substrate after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM412610(1-(2-((2-ethoxy-4-(4-methyl-4H-1,2,4-triazol-3-yl)...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104371(US8575186, 134/183/184 | US8575186, 199 | US857518...)
Affinity DataKi:  0.260nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104331(US8575186, 177 | US8575186, 178 | US8575186, 94/16...)
Affinity DataKi:  0.280nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104408(US8575186, 171/172 | US8575186, 188)
Affinity DataKi:  0.280nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104378(US8575186, 141)
Affinity DataKi:  0.290nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104382(US8575186, 145)
Affinity DataKi:  0.310nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104467(US8575186, 230/231 | US8575186, 247)
Affinity DataKi:  0.310nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364980(CHEMBL1950775)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364980(CHEMBL1950775)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104331(US8575186, 177 | US8575186, 178 | US8575186, 94/16...)
Affinity DataKi:  0.320nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104361(US8575186, 124)
Affinity DataKi:  0.330nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364981(CHEMBL1950776)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104371(US8575186, 134/183/184 | US8575186, 199 | US857518...)
Affinity DataKi:  0.350nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104477(US8575186, 240/241 | US8575186, 257)
Affinity DataKi:  0.350nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364981(CHEMBL1950776)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364981(CHEMBL1950776)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104408(US8575186, 171/172 | US8575186, 188)
Affinity DataKi:  0.360nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364980(CHEMBL1950775)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104331(US8575186, 177 | US8575186, 178 | US8575186, 94/16...)
Affinity DataKi:  0.370nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50464038(CHEMBL4250961)
Affinity DataKi:  0.380nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104402(US8575186, 165/166 | US8575186, 182)
Affinity DataKi:  0.410nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104321(US8575186, 250 | US8575186, 251 | US8575186, 84/23...)
Affinity DataKi:  0.420nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104371(US8575186, 134/183/184 | US8575186, 199 | US857518...)
Affinity DataKi:  0.420nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104475(US8575186, 238/239 | US8575186, 255)
Affinity DataKi:  0.430nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM241226(US10479788, Example 68 | US11046688, Example 68 | ...)
Affinity DataKi:  0.440nMAssay Description:Inhibition of full length human N-terminal 6xHis-tagged MPS1 expressed in baculovirus expression system using 5FAM-H236 peptide as substrate after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104454(US8575186, 217/218 | US8575186, 234)
Affinity DataKi:  0.460nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104376(US8575186, 139)
Affinity DataKi:  0.470nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104360(US8575186, 123)
Affinity DataKi:  0.470nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104302(US8575186, 203 | US8575186, 204 | US8575186, 65/18...)
Affinity DataKi:  0.5nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM241226(US10479788, Example 68 | US11046688, Example 68 | ...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of human full length MPS1 expressed in recombinant baculovirus infected Sf9 insect cells using 5FAM-DHTGFLTEYVATRCONH2 as substrate after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104430(US8575186, 193/194 | US8575186, 210)
Affinity DataKi:  0.5nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104456(US8575186, 219/220 | US8575186, 236)
Affinity DataKi:  0.5nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104446(US8575186, 209/215/216 | US8575186, 231 | US857518...)
Affinity DataKi:  0.530nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104462(US8575186, 225/226 | US8575186, 242)
Affinity DataKi:  0.530nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104377(US8575186, 140)
Affinity DataKi:  0.560nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104458(US8575186, 221/222 | US8575186, 238)
Affinity DataKi:  0.560nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104320(US8575186, 228 | US8575186, 229 | US8575186, 83/21...)
Affinity DataKi:  0.570nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104479(US8575186, 242/243 | US8575186, 259)
Affinity DataKi:  0.580nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104302(US8575186, 203 | US8575186, 204 | US8575186, 65/18...)
Affinity DataKi:  0.590nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Displayed 1 to 50 (of 2081 total ) | Next | Last >>
Jump to: