Affinity DataKi: 0.313nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Pharmaceutical Research Center
Curated by ChEMBL
Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity for 5-hydroxytryptamine 3 receptor was determined by measuring displacement of [3H]GR-65630 from rat brain corticesMore data for this Ligand-Target Pair
Affinity DataKi: 0.534nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Pharmaceutical Research Center
Curated by ChEMBL
Pharmaceutical Research Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity for 5-hydroxytryptamine 3 receptor was determined by measuring displacement of [3H]GR-65630 from rat brain corticesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 119nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 248nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 588nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 695nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.41E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.41E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.88E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.41E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.95E+3nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.02E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.82E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.54E+4nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.96E+4nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.98E+4nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.36E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.98E+4nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.47E+4nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.83E+4nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.76E+4nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.31E+5nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+6nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair