TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.530nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.660nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.660nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human TACE by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of human FLT D835Y mutant using 10 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of human FLT3 using 10 uM ATPMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human TNF-alpha by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of IKKbeta kinase (unknown origin) by Lance ULight systemMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of FLT3 kinase (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of human FLT3 using 10 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human TNF-alpha by fluorescent spectroscopyMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of FLT3 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of FLT3 kinase (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of human FLT3 using 10 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using Fluor de Lys as substrate incubated with compound for 30 mins by microtiter-plate reading...More data for this Ligand-Target Pair