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Found 86 with Last Name = 'yang' and Initial = 'sx'
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50118955(CHEMBL94678 | Compound K-252a(epi))
Affinity DataIC50:  1.20nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50410231(CHEMBL2113064)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50410233(CHEMBL2113063)
Affinity DataIC50:  3nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50167984(CHEMBL370493 | K-252a analogue)
Affinity DataIC50:  4nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50167984(CHEMBL370493 | K-252a analogue)
Affinity DataIC50:  4nMAssay Description:Inhibition of baculovirus expressed human VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50167983(CHEMBL365585 | K-252a analogue)
Affinity DataIC50:  4nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50118955(CHEMBL94678 | Compound K-252a(epi))
Affinity DataIC50:  5nMAssay Description:Inhibition of NGF-stimulated TrkA phosphorylation in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203095(4-((4-bromo-5-methoxy-1-methyl-1H-indol-3-yl)methy...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182149(4-((4-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(p...)
Affinity DataIC50:  6nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50377290(CHEMBL427901)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant TrkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203075(4-((4-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(1...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182139(4-((4-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  9nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50377300(CHEMBL254555)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant TrkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203079(4-((4,7-dimethoxy-1-methyl-1H-indol-3-yl)methylene...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182144(4-((5-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  10nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203103(4-((4-bromo-1,6-dimethyl-1H-indol-3-yl)methylene)-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
Affinity DataIC50:  13nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203106(4-((4-methoxy-1-methyl-1H-indol-3-yl)methylene)-3-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50377298(CHEMBL404561)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant TrkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203085(4-((4-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203097(4-((4-fluoro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203074(4-((4-ethoxy-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  16nMAssay Description:Inhibition of VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182141(4-((4-fluoro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  17nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182152(4-((5-methyl-5H-[1,3]dioxolo[4,5-f]indol-7-yl)meth...)
Affinity DataIC50:  17nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203091(4-((4-methoxy-1-methyl-1H-indol-3-yl)methylene)-3-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203074(4-((4-ethoxy-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  19nMAssay Description:Inhibition of FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203098(4-((4,7-dimethoxy-1-methyl-1H-indol-3-yl)methylene...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50410232(CHEMBL2113062)
Affinity DataIC50:  20nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203089(CHEMBL398459 | methyl 1-methyl-3-((5-oxo-3-(1,2,3-...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182151(4-((5-fluoro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  23nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203109(4-((4-bromo-5-methoxy-1-methyl-1H-indol-3-yl)methy...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203108(4-((4-ethoxy-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182146(4-((4-methoxy-1-methyl-1H-indol-3-yl)methylene)-3-...)
Affinity DataIC50:  26nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203078(4-((5-methoxy-1-methyl-1H-indol-3-yl)methylene)-3-...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50410234(CHEMBL2113065)
Affinity DataIC50:  29nMAssay Description:Inhibition of baculovirus expressed human trkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182140(4-((5-methoxy-1-methyl-1H-indol-3-yl)methylene)-3-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182142(4-((5-methyl-5H-[1,3]dioxolo[4,5-f]indol-7-yl)meth...)
Affinity DataIC50:  32nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50377299(CHEMBL404385)
Affinity DataIC50:  33nMAssay Description:Inhibition of human recombinant TrkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203093(4-((5-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203090(4-((4-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(4...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203077(4-((1,5-dimethyl-1H-indol-3-yl)methylene)-3-(1,2,3...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203074(4-((4-ethoxy-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  36nMAssay Description:Inhibition of TRK AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50155151(4-((1-methyl-1H-indol-3-yl)methylene)-3-(pyrazin-2...)
Affinity DataIC50:  37nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203074(4-((4-ethoxy-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182137(4-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)-3-(pyra...)
Affinity DataIC50:  43nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50377295(CHEMBL402067)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant TrkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203099(4-((4-chloro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182148(4-((4-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(t...)
Affinity DataIC50:  45nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50182136(4-((1-methyl-1H-indol-3-yl)methylene)-3-(thiazol-2...)
Affinity DataIC50:  46nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203082(4-((5-fluoro-1-methyl-1H-indol-3-yl)methylene)-3-(...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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