Affinity DataKi: 9.10nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding Affinity towards Adenosine A2A receptor expressed in HEK-293 cells versus [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding Affinity for adenosine A2A receptor expressed in HEK-293 cells compared to [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding Affinity for adenosine A2A receptor expressed in HEK-293 cells compared to [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity towards adenosine A3 receptor expressed in HEK-293 cells versus [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding Affinity for adenosine A2A receptor expressed in HEK-293 cells compared to [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.00500nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.0100nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.0100nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.0400nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.0710nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against cyclic AMP production in rat Adenosine A2A receptor assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibitory activity on NECA-induced cyclic-AMP accumulation in CHO-K1 cells expressing human Adenosine A2B receptorMore data for this Ligand-Target Pair