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Found 108 with Last Name = 'zalkow' and Initial = 'lh'
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005897(CHEMBL40840 | Carbonic acid 8-butoxycarbonyloxy-3-...)
Affinity DataKi:  150nMAssay Description:HLE-inhibitor (Human Leukocyte Elastase) dissociation constant determined by using Dixon PlotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005903(CHEMBL44123 | Carbonic acid 8-butoxycarbonyloxy-7-...)
Affinity DataKi:  430nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005900(CHEMBL43983 | Carbonic acid 8-butoxycarbonyloxy-3-...)
Affinity DataKi:  1.90E+3nMAssay Description:HLE-inhibitor (Human Leukocyte Elastase) dissociation constant determined by using Dixon PlotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005887(CHEMBL440290 | Carbonic acid 8-butoxycarbonyloxy-6...)
Affinity DataKi:  2.80E+3nMAssay Description:HLE-inhibitor (Human Leukocyte Elastase) dissociation constant determined by using Dixon PlotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005889(CHEMBL40878 | Carbonic acid 8-butoxycarbonyloxy-9,...)
Affinity DataKi:  7.50E+3nMAssay Description:HLE-inhibitor (Human Leukocyte Elastase) dissociation constant determined by using Dixon PlotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097532(CHEMBL354794 | [17-(1,5-Dimethyl-hexyl)-10,13-dime...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Howard University

Curated by ChEMBL
LigandPNGBDBM50308752(3-(1-tert-butyl-4-amino-1H-pyrazolo[3,4-d]pyrimidi...)
Affinity DataIC50:  759nMAssay Description:Inhibition of CBR-mediated NADPH-dependent reduction of menadione to menadiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Howard University

Curated by ChEMBL
LigandPNGBDBM50308752(3-(1-tert-butyl-4-amino-1H-pyrazolo[3,4-d]pyrimidi...)
Affinity DataIC50:  788nMAssay Description:Inhibition of CBR-mediated NADPH-dependent reduction of menadione to menadiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097529(CHEMBL354215 | [17-(1,5-Dimethyl-hexyl)-10,13-dime...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097528(CHEMBL169020 | Dithiocarbonic acid O-[17-(1,5-dime...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005895(CHEMBL416614 | Carbonic acid 4,5-bis-butoxycarbony...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005897(CHEMBL40840 | Carbonic acid 8-butoxycarbonyloxy-3-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005903(CHEMBL44123 | Carbonic acid 8-butoxycarbonyloxy-7-...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097542(CHEMBL354816 | Phenyl-thiocarbamic acid O-[17-(1,5...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097530(CHEMBL168868 | [5-(5-Cyano-1-methyl-pentyl)-1-(1,5...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50068031(CHEMBL142455 | [(1R,3aS,4R,5S,7aR)-5-(5-Cyano-1-me...)
Affinity DataIC50:  2.20E+3nMAssay Description:Compound was evaluated for the inhibition of Cdc25A phosphatase by using fluorescein diphosphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097530(CHEMBL168868 | [5-(5-Cyano-1-methyl-pentyl)-1-(1,5...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50068031(CHEMBL142455 | [(1R,3aS,4R,5S,7aR)-5-(5-Cyano-1-me...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097539(CHEMBL354578 | [5-(5-Cyano-1-methyl-pent-1-enyl)-1...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005887(CHEMBL440290 | Carbonic acid 8-butoxycarbonyloxy-6...)
Affinity DataIC50:  2.50E+3nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097526(CHEMBL172392 | [5-(5-Cyano-4-ethoxy-1-methylene-pe...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Howard University

Curated by ChEMBL
LigandPNGBDBM50308753(3-(Methyl-N-ethylcarbamate)-5-hydroxybenz[f]indazo...)
Affinity DataIC50:  3.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005883(1,8-Dihydroxy-2-pentyl-anthraquinone | CHEMBL40884)
Affinity DataIC50:  3.90E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Howard University

Curated by ChEMBL
LigandPNGBDBM50308751(3-(methyl-N-ethylcarbamate)-6-(N0-ethylphenylamino...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Howard University

Curated by ChEMBL
LigandPNGBDBM50308750(3-(Methyl-N-ethylcarbamate)-6-(N0-methylphenylamin...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50068037(5-(Benzoyl-{2-[(2,5-diphenyl-oxazole-4-carbonyl)-a...)
Affinity DataIC50:  4.00E+3nMAssay Description:Compound was evaluated for the inhibition of Cdc25A phosphatase by using p-nitrophenylphosphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005884(2-Hexyl-1,8-dihydroxy-anthraquinone | CHEMBL41317)
Affinity DataIC50:  4.20E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005882(1,8-Dihydroxy-2-propyl-anthraquinone | CHEMBL40292)
Affinity DataIC50:  4.20E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Howard University

Curated by ChEMBL
LigandPNGBDBM50308754(3-(Methyl-N-ethylcarbamate)-6,7-dichloro-5,8-dimet...)
Affinity DataIC50:  5.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097534(5-[3-(1,5-Dimethyl-hexyl)-3a,6-dimethyl-8-oxo-dode...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005900(CHEMBL43983 | Carbonic acid 8-butoxycarbonyloxy-3-...)
Affinity DataIC50:  5.10E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097540(CHEMBL434693 | [1-(1,5-Dimethyl-hexyl)-7a-methyl-5...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005898(1,8-Dihydroxy-3-methyl-6-propoxy-anthraquinone | C...)
Affinity DataIC50:  5.90E+3nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte Elastase (HLE) at 62 uM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005905(2-Butyl-1-hydroxy-8-methoxy-anthraquinone | CHEMBL...)
Affinity DataIC50:  5.90E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097544(CHEMBL169414 | [1-(1,5-Dimethyl-hexyl)-7a-methyl-5...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005885(2-Hexyl-1-hydroxy-8-methoxy-anthraquinone | CHEMBL...)
Affinity DataIC50:  6.00E+3nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005888(1-Hydroxy-8-methoxy-2-pentyl-anthraquinone | CHEMB...)
Affinity DataIC50:  6.10E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005886(1,8-Dihydroxy-3-methoxy-6-methylanthraquinone | 1,...)
Affinity DataIC50:  6.20E+3nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte Elastase (HLE) at 65 uM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005896(2-Butyl-1,8-dihydroxy-anthraquinone | CHEMBL41504)
Affinity DataIC50:  6.40E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 3(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50068031(CHEMBL142455 | [(1R,3aS,4R,5S,7aR)-5-(5-Cyano-1-me...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibitory activity tested against Human cell division cycle 25 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005902(2-Benzyl-1-hydroxy-anthraquinone | CHEMBL43177)
Affinity DataIC50:  6.60E+3nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005915(2-Benzyl-1-hydroxy-8-methoxy-anthraquinone | CHEMB...)
Affinity DataIC50:  6.70E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097546(Sulfuric acidmono-{5-furan-3-yl-2-methyl-1-[1-(2,5...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005891(1,8-Dihydroxy-2-isobutyl-anthraquinone | CHEMBL434...)
Affinity DataIC50:  8.00E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division control protein 45 homolog(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097530(CHEMBL168868 | [5-(5-Cyano-1-methyl-pentyl)-1-(1,5...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibitory activity tested against human cell division cycle 45-like 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50005892(1-Hydroxy-8-methoxy-2-propyl-anthraquinone | CHEMB...)
Affinity DataIC50:  8.70E+3nMAssay Description:In vitro inhibition of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097530(CHEMBL168868 | [5-(5-Cyano-1-methyl-pentyl)-1-(1,5...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibitory activity tested against Human CD45 Phosphatase (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50097543(CHEMBL165813 | [5-(4-Acetoxy-1-methyl-2-oxo-cycloh...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50341997(CHEMBL1765353 | Dysidiolide)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibitory activity tested against cell division cycle 25A (assay using fluorescein diphosphate (FDP) as substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50341997(CHEMBL1765353 | Dysidiolide)
Affinity DataIC50:  9.40E+3nMAssay Description:Compound was evaluated for the inhibition of Cdc25A phosphatase by using p-nitrophenylphosphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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