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Found 13 with Last Name = 'zappelli' and Initial = 'e'
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341243((3S,6R)-1-[6-(3-Amino-1H-indazol-6-yl)-2-(methylam...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of PDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590814(CHEMBL5182359)
Affinity DataIC50:  6nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590815(CHEMBL5199785)
Affinity DataIC50:  11nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590813(CHEMBL5204846)
Affinity DataIC50:  17nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590815(CHEMBL5199785)
Affinity DataIC50:  18nMAssay Description:Inhibition of MDM4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590813(CHEMBL5204846)
Affinity DataIC50:  25nMAssay Description:Inhibition of MDM4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50184998(CHEMBL3823242)
Affinity DataIC50:  27nMAssay Description:Inhibition of PDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590814(CHEMBL5182359)
Affinity DataIC50:  27nMAssay Description:Inhibition of MDM4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50185001(CHEMBL3824119 | US10351548, Compound IB35)
Affinity DataIC50:  112nMAssay Description:Inhibition of PDK1 (unknown origin) by FRET-based Z-lyte assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50185000(CHEMBL3823844 | US10351548, Compound SA16)
Affinity DataIC50:  416nMAssay Description:Inhibition of PDK1 (unknown origin) by FRET-based Z-lyte assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50185003(CHEMBL3824264 | US10351548, Compound JJ31)
Affinity DataIC50:  512nMAssay Description:Inhibition of PDK1 (unknown origin) by FRET-based Z-lyte assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50184999(CHEMBL3823622 | US10351548, Compound SA23)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of PDK1 (unknown origin) by FRET-based Z-lyte assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50185002(CHEMBL3822974 | US10351548, Compound IB32)
Affinity DataIC50:  6.68E+3nMAssay Description:Inhibition of PDK1 (unknown origin) by FRET-based Z-lyte assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed