TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 680nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.02E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.03E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.14E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.19E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.28E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.36E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.42E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.49E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.87E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 2.26E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 2.36E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 2.77E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 2.78E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 3.68E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 3.68E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 6.33E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 6.74E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 8.35E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition of recombinant HIV-1 integrase strand transfer activity using 32P 5' end-labeled linear 21'mer as substrate preincubated for 30 mins prior...More data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of His6-tagged HIV-1 integrase assessed as decrease in integrase-Flag-LEDGF/p75 interaction preincubated with enzyme for 30 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant HIV-1 integrase strand transfer activity using 32P 5' end-labeled linear 21'mer as substrate preincubated for 30 mins prior...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair