TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human platelet COX1 by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 790nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 5.71E+3nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in glucose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Oryctolagus cuniculus (rabbit))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of 15LOX in rabbit reticulocytes by EIA assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in glucose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.44E+4nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 2.86E+4nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 7.39E+4nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: 9.02E+4nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human platelet COX1 by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells by EIA assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tahitian Noni International
Curated by ChEMBL
Tahitian Noni International
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of 5LOX in human PBMC by EIA assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: >2.01E+5nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in glucose medium by microtiter plate assayMore data for this Ligand-Target Pair