BindingDB PrimarySearch_ki

Found 226 with Last Name = 'zhou' and Initial = 'k'

Cocaine esterase(Homo sapiens (Human))
Dalian Institute Of Chemical Physics

Curated by ChEMBL

PNG

BDBM50154561(CHEMBL3774603)

Ki: 42nMAssay Description:Competitive inhibition of CE2 in human liver microsomes using fluorescein diacetate as substrate preincubated for 10 mins followed by substrate addit...More data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Cocaine esterase(Homo sapiens (Human))
Dalian Institute Of Chemical Physics

Curated by ChEMBL

PNG

BDBM50130903(CHEMBL3632950)

Ki: 1.76E+3nMAssay Description:Fixed inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by Dixon and Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609320(CHEMBL5272699)

IC50: 0.650nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609337(CHEMBL5270700)

IC50: 0.780nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609315(CHEMBL5274219)

IC50: 0.920nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609339(CHEMBL5271782)

IC50: 1.10nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609333(CHEMBL5291238)

IC50: 1.10nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609307(CHEMBL5288947)

IC50: 1.60nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details PubMed PDB

3D Structure (crystal)

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609313(CHEMBL5283756)

IC50: 2.30nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609334(CHEMBL5287824)

IC50: 2.5nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609318(CHEMBL5271800)

IC50: 2.90nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609306(CHEMBL5289496)

IC50: 3.70nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609300(CHEMBL5266562)

IC50: 3.70nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details PubMed PDB

3D Structure (crystal)

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609322(CHEMBL5284876)

IC50: 3.80nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609319(CHEMBL5289683)

IC50: 3.80nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM440444(US10633389, Example 109-3 | US20230279020, Example...)

IC50: 3.80nMAssay Description:Inhibition of FLAG-tagged CARM1 (unknown origin) (2 to 585 residues) using biotin-aminohexanoate-PRKQLATKAARMeKSAP-amide peptide as substrate preincu...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Purchase PC cid PC sid PDB

Details PubMed PDB

3D Structure (crystal)

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609332(CHEMBL5268692)

IC50: 4.20nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609317(CHEMBL5274541)

IC50: 4.30nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609324(CHEMBL5277620)

IC50: 4.40nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609312(CHEMBL5273938)

IC50: 5.10nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609311(CHEMBL5279093)

IC50: 5.20nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM440444(US10633389, Example 109-3 | US20230279020, Example...)

IC50: 6nMAssay Description:Inhibition of FLAG-tagged CARM1 (unknown origin) (2 to 585 residues) using biotin-aminohexanoate-PRKQLATKAARMeKSAP-amide peptide as substrate preincu...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Purchase PC cid PC sid PDB

Details PubMed PDB

3D Structure (crystal)

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609323(CHEMBL5290292)

IC50: 6.10nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609316(CHEMBL5269937)

IC50: 6.20nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606107(CHEMBL5169557)

IC50: 8nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609305(CHEMBL5290611)

IC50: 10nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609301(CHEMBL4559961)

IC50: <10nMAssay Description:Inhibition of FLAG-tagged CARM1 (unknown origin) (2 to 585 residues) using biotin-aminohexanoate-PRKQLATKAARMeKSAP-amide peptide as substrate preincu...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details PubMed PDB

3D Structure (crystal)

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609340(CHEMBL5289773)

IC50: 10nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606116(CHEMBL5187366)

IC50: 10nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606105(CHEMBL5208750)

IC50: 11nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609336(CHEMBL5285757)

IC50: 12nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609321(CHEMBL5266548)

IC50: 12nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606106(CHEMBL5204119)

IC50: 12nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609341(CHEMBL5270405)

IC50: 12nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609335(CHEMBL5279447)

IC50: 13nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606108(CHEMBL5196712)

IC50: 14nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606117(CHEMBL5188230)

IC50: 17nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606119(CHEMBL5205007)

IC50: 17nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Cocaine esterase(Homo sapiens (Human))
Dalian Institute Of Chemical Physics

Curated by ChEMBL

PNG

BDBM50154561(CHEMBL3774603)

IC50: 20nMAssay Description:Inhibition of CE2 in human liver microsomes using fluorescein diacetate as substrate preincubated for 10 mins followed by substrate addition measured...More data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609342(CHEMBL5271681)

IC50: 20nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone deacetylase 6(Homo sapiens (Human))
Fudan University

Curated by ChEMBL

PNG

BDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)

IC50: 21nMAssay Description:Inhibition of recombinant HDAC6 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609326(CHEMBL5287686)

IC50: 21nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606129(CHEMBL5179194)

IC50: 22nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM177922(US10307413, Compound 337 | US10391089, Compound 16...)

IC50: 22nMAssay Description:Inhibition of PRMT5 (unknown origin) by biochemical assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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3D Structure (crystal)

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50609338(CHEMBL5289833)

IC50: 22nMAssay Description:Inhibition of human CARM1 (140 to 480 residues) incubated for 15 mins measured after 60 min by AlphaLISA assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606115(CHEMBL5177256)

IC50: 22nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606118(CHEMBL5176474)

IC50: 22nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606100(CHEMBL5173004)

IC50: 24nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Purchase PC cid PC sid

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL

PNG

BDBM50606135(CHEMBL5178858)

IC50: 24nMAssay Description:Displacement of [3H]-SAM from PRMT5 (unknown origin) using peptide substrate preincubated for 15 mins followed by substrate addition for 60 mins by r...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))TBA

PNG

BDBM50532879(CHEMBL3347611)

IC50: 27nMAssay Description:Inhibition of FLAG-tagged CARM1 (unknown origin) (2 to 585 residues) using biotin-aminohexanoate-PRKQLATKAARMeKSAP-amide peptide as substrate preincu...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

KEGG PC cid PC sid

Displayed 1 to 50 (of 226 total ) | Next | Last >>

Filter my 226 hits

Targets 23▿
- Histone-arginine methyltransferase CARM1 47
- Cocaine esterase 42
- Protein arginine N-methyltransferase 5 40
- Histone acetyltransferase p300 32
- Nuclear receptor ROR-gamma 18
- Liver carboxylesterase 1 17
- Beta-glucuronidase 5
- Capsid protein 3
- Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 2
- Histone deacetylase 8 2
- Histone deacetylase 6 2
- Histone deacetylase 2 2
- Histone deacetylase 3 2
- Histone deacetylase 1 2
- Protein arginine N-methyltransferase 1 2
- Histone-lysine N-methyltransferase 2A 1
- Histone-lysine N-methyltransferase 2B 1
- Protein arginine N-methyltransferase 6 1
- Protein arginine N-methyltransferase 7 1
- Protein arginine N-methyltransferase 8 1
- Histone-lysine N-methyltransferase NSD2 1
- Histone-lysine N-methyltransferase EZH2 1
- Protein arginine N-methyltransferase 3 1
- ...
Publications 8▿
- J Med Chem 65: 7854-7875 (2022) 45
- Eur J Med Chem 180: 171-190 (2019) 42
- Eur J Med Chem 112: 280-8 (2016) 35
- J Nat Prod 78: 2372-80 (2015) 24
- Eur J Med Chem 187: (2020) 18
- J Nat Prod 83: 825-833 (2020) 5
- ACS Med Chem Lett 8: 969-974 (2017) 3
- Bioorg Med Chem 27: 2235-2244 (2019) 2
Institutions 7▿
- Fudan University 60
- Sun Yat-Sen University 45
- Dalian Institute Of Chemical Physics 35
- Liaoning University Of Traditional Chinese Medicine 24
- Wayne State University 5
- Wuxi Apptec (Shanghai) 3
- Sichuan University 2
Affinity: 0.65 to 1.0E+5 nM▿
- Ki 2
- IC50 223
- EC50 1
- Affinity ≤ nM
Xtal structures: 6
Docked structures: 1
Catalog Cmpds: 21