TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University
Curated by ChEMBL
Fourth Military Medical University
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University
Curated by ChEMBL
Fourth Military Medical University
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University
Curated by ChEMBL
Fourth Military Medical University
Curated by ChEMBL
Affinity DataIC50: 1.48nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University
Curated by ChEMBL
Fourth Military Medical University
Curated by ChEMBL
Affinity DataIC50: 3.62nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University
Curated by ChEMBL
Fourth Military Medical University
Curated by ChEMBL
Affinity DataIC50: 8.14nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University
Curated by ChEMBL
Fourth Military Medical University
Curated by ChEMBL
Affinity DataIC50: 17.6nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant N-terminal 6his-tagged BRD4 expressed in Escherichia coli BL21(DE3) using H4 peptide as substrate by alphascreen assa...More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD4 bromodomain (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant N-terminal 6his-tagged BRD4 bromodomain 2 expressed in Escherichia coli BL21(DE3) using using H4 peptide as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 722nMAssay Description:Activation of human P2Y1 receptor expressed in human 1321N1 cells assessed as induction of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 10.3nMAssay Description:Activation of human P2Y1 receptor expressed in human 1321N1 cells assessed as induction of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.89nMAssay Description:Agonist activity at human P2Y1 receptor expressed in human 1321N1 cells by PLC assayMore data for this Ligand-Target Pair