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Found 26 with Last Name = 'zhou' and Initial = 'sy'
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50306490((+)-(S)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50:  0.420nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50:  0.760nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50306490((+)-(S)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50:  1.48nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50:  3.62nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50:  8.14nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50:  17.6nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human recombinant N-terminal 6his-tagged BRD4 expressed in Escherichia coli BL21(DE3) using H4 peptide as substrate by alphascreen assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)
Affinity DataIC50:  90nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)
Affinity DataIC50:  220nMAssay Description:Inhibition of BRD4 bromodomain (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataIC50:  510nMAssay Description:Inhibition of human recombinant N-terminal 6his-tagged BRD4 bromodomain 2 expressed in Escherichia coli BL21(DE3) using using H4 peptide as substrate...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525654(CHEMBL4533819)
Affinity DataIC50:  550nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525650(CHEMBL4592461)
Affinity DataIC50:  800nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525648(CHEMBL4471181)
Affinity DataIC50:  860nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525647(CHEMBL4456714)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525657(CHEMBL4581142)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525656(CHEMBL4527844)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525649(CHEMBL4555713)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525652(CHEMBL4472855)
Affinity DataIC50:  1.81E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525655(CHEMBL4460102)
Affinity DataIC50:  1.81E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525653(CHEMBL4461915)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525646(CHEMBL4582953)
Affinity DataIC50:  1.96E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525651(CHEMBL4470171)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50525658(CHEMBL4574735)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50308552((1'S,2'R,3'S,4'R,5'S)-4-(6-Amino-2-chloro-9H-purin...)
Affinity DataEC50:  722nMAssay Description:Activation of human P2Y1 receptor expressed in human 1321N1 cells assessed as induction of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50118242(((2R,3S,4R,5R)-5-(6-amino-2-(methylthio)-9H-purin-...)
Affinity DataEC50:  10.3nMAssay Description:Activation of human P2Y1 receptor expressed in human 1321N1 cells assessed as induction of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50308552((1'S,2'R,3'S,4'R,5'S)-4-(6-Amino-2-chloro-9H-purin...)
Affinity DataEC50:  1.89nMAssay Description:Agonist activity at human P2Y1 receptor expressed in human 1321N1 cells by PLC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed