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Found 132 with Last Name = 'zomaya' and Initial = 'a'
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113399(4-[2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-phenyl-...)
Affinity DataKi:  423nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113373(2-Cyclopentyloxy-4-(1,2-diphenyl-ethyl)-1-methoxy-...)
Affinity DataKi:  1.17E+3nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113366(4-[2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-phenyl-...)
Affinity DataKi: >8.00E+3nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113362(1-{3-[1-((R)-3-Cyclopentyloxy-4-methoxy-phenyl)-2-...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114291((S)-2-[(3,5-Dichloro-pyridine-4-carbonyl)-amino]-3...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of VLA-4 expressed in Jurkat cell line, in a cell-based adhesion assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114276((S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amin...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of VLA-4 from HL60 lysate in a protein-based ligand binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114276((S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amin...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of VLA-4 from HL60 lysate in a protein-based ligand binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113380(4-{(R)-2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-[4-...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114291((S)-2-[(3,5-Dichloro-pyridine-4-carbonyl)-amino]-3...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of VLA-4 from HL60 lysate in a protein-based ligand binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114316((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  1nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114300(3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino]-ph...)
Affinity DataIC50:  2nMAssay Description:Inhibition of very late antigen 4 from HL60 lysate in a protein-based ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114296((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  2nMAssay Description:Inhibition of very late antigen 4 from HL60 lysate in a protein-based ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113389(CHEMBL285766 | N-{4-[(R)-1-(3-Cyclopentyloxy-4-met...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113372(4-[(S)-2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-thi...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114298(2-[5-Chloro-4-(propane-1-sulfonyl)-pyridin-2-ylami...)
Affinity DataIC50:  4nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114301((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  4nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114310(6-((S)-1-Carboxy-2-{4-[(3,5-dichloro-pyridine-4-ca...)
Affinity DataIC50:  4nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113377(1-{4-[(R)-1-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50064858((R)-4-(2-(3-(cyclopentyloxy)-4-methoxyphenyl)-2-ph...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113363(CHEMBL286921 | N-{4-[(R)-1-(3-Cyclopentyloxy-4-met...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113390(CHEMBL286118 | Pyrrolidine-1-carboxylic acid {3-[(...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113381(4-[(R)-1-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-pyr...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113378(4-[(S)-2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-fur...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114305((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  6nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114295((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  6nMAssay Description:Inhibition of very late antigen 4 from HL60 lysate in a protein-based ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114292(1-[4-((S)-1-Carboxy-2-{4-[(3,5-dichloro-pyridine-4...)
Affinity DataIC50:  6nMAssay Description:Inhibition of VLA-4 expressed in Jurkat cell line, in a cell-based adhesion assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113392(CHEMBL36559 | N-{4-[(R)-1-(3-Cyclopentyloxy-4-meth...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113386(CHEMBL35011 | Propane-2-sulfonic acid {4-[(R)-1-(3...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113387(4-[(R)-2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-phe...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114277((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  7nMAssay Description:Inhibition of VLA-4 from HL60 lysate in a protein-based ligand binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114299((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  7nMAssay Description:Inhibition of very late antigen 4 from HL60 lysate in a protein-based ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114297(2-[5-Chloro-4-(propane-1-sulfinyl)-pyridin-2-ylami...)
Affinity DataIC50:  7nMAssay Description:Inhibition of very late antigen 4 from HL60 lysate in a protein-based ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113369(CHEMBL286421 | N-{4-[(R)-1-(3-Cyclopentyloxy-4-met...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113391(CHEMBL287359 | N-{4-[(R)-1-(3-Cyclopentyloxy-4-met...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114280((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  8nMAssay Description:Inhibition of VLA-4 from HL60 lysate in a protein-based ligand binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113404(4-[2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-(3-fluo...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113396(4-[(R)-2-(3-cyclopentyloxy-4-methoxy-phenyl)-2-pyr...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113364(CHEMBL416399 | N-(methylsulfonyl)-N-[4-(1-{3-cyclo...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114311(6-(1-Carboxy-2-{4-[(3,5-dichloro-pyridine-4-carbon...)
Affinity DataIC50:  10nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114315((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  10nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113371(CHEMBL289012 | Pyrrolidine-1-carboxylic acid {4-[(...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113385(3-{4-[(R)-1-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113367(CHEMBL287167 | N,N-dimethyl-N'-{3-[(1S)-1-{3-cyclo...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114289((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  14nMAssay Description:Inhibition of VLA-4 expressed in Jurkat cell line, in a cell-based adhesion assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114307(6-((S)-1-Carboxy-2-{4-[(3,5-dichloro-pyridine-4-ca...)
Affinity DataIC50:  14nMAssay Description:Inhibition of very late antigen 4 expressed in Jurkat cell line, in a cell-based adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113401(3-{3-[(R)-1-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50114288((S)-3-{4-[(3,5-Dichloro-pyridine-4-carbonyl)-amino...)
Affinity DataIC50:  16nMAssay Description:Inhibition of VLA-4 expressed in Jurkat cell line, in a cell-based adhesion assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113361(4-[2-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-(4-meth...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113382(4-(2-(3-(cyclopentyloxy)-4-methoxyphenyl)-2-phenyl...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113393(1-{3-[1-((R)-3-Cyclopentyloxy-4-methoxy-phenyl)-2-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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