Affinity DataIC50: 300nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of HIV 1 integrase strand transfer activityMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processing was tested in CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein(Rous sarcoma virus (strain Prague C) (RSV-PrC))
Cnrs Umr 8532
Curated by ChEMBL
Cnrs Umr 8532
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein(Rous sarcoma virus (strain Prague C) (RSV-PrC))
Cnrs Umr 8532
Curated by ChEMBL
Cnrs Umr 8532
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.Checked by AuthorMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Cnrs Umr 8532
Curated by ChEMBL
Cnrs Umr 8532
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Compound was tested in vitro to inhibit human immuno virus-1 (HIV-1) using enzymatic disintegration assay.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer (integration)More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Cnrs Umr 8532
Curated by ChEMBL
Cnrs Umr 8532
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Compound was tested in vitro to inhibit human immuno virus-1 (HIV-1) using enzymatic disintegration assay.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Cnrs Umr 8532
Curated by ChEMBL
Cnrs Umr 8532
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Compound was tested in vitro to inhibit human immuno virus-1 (HIV-1) using enzymatic disintegration assay.Checked by AuthorMore data for this Ligand-Target Pair