Affinity DataIC50: 4.5nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of glyceraldehyde reduction activity of human AKR1B1More data for this Ligand-Target Pair
Affinity DataIC50: 11.4nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B10(Homo sapiens (Human))
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of retinaldehyde reductase activity of human AKR1B10More data for this Ligand-Target Pair
Affinity DataIC50: 13.7nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Inverse agonist activity at RARalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 161nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Antagonist activity at yeast GAL4 fused mouse RARalpha ligand binding domain expressed in HeLa cells assessed as inhibition of TTNPB-induced receptor...More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Antagonist activity at yeast GAL4 fused mouse RARbeta ligand binding domain expressed in HeLa cells assessed as inhibition of TTNPB-induced receptor ...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat AKR1B4More data for this Ligand-Target Pair
Affinity DataIC50: 1.28E+3nMAssay Description:Antagonist activity at Gal4-fused RARalpha (unknown origin) transfected in HEK293 cells assessed as inhibition of ATRA-induced transcriptional activi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at yeast GAL4 fused mouse RARbeta ligand binding domain expressed in HeLa cells assessed as inhibition of TTNPB-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.65E+3nMAssay Description:Antagonist activity at Gal4-fused RARalpha (unknown origin) transfected in HEK293 cells assessed as inhibition of ATRA-induced transcriptional activi...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at yeast GAL4 fused mouse RARgamma ligand binding domain expressed in HeLa cells assessed as inhibition of TTNPB-induced receptor...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 3.37E+3nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 4.43E+3nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.47E+3nMAssay Description:Antagonist activity at Gal4-fused RARalpha (unknown origin) transfected in HEK293 cells assessed as inhibition of ATRA-induced transcriptional activi...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 4.75E+3nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 5.16E+3nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of purified recombinant histidine-HA-tagged IKKbeta (unknown origin) expressed in SF9 cellsMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 7.06E+3nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 7.81E+3nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at yeast GAL4 fused mouse RARgamma ligand binding domain expressed in HeLa cells assessed as inhibition of TTNPB-induced receptor...More data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of human DNMT1 using AdoMet and poly dI-dC after 2 hrs by radioactive assayMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC4More data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Dissociation constant for binding to Retinoic acid receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 50nMAssay Description:Dissociation constant for binding to Retinoic acid receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Dissociation constant for binding to Retinoic acid receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 60nMAssay Description:Dissociation constant for Retinoid X receptor alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKd: 26nMAssay Description:Dissociation constant for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKd: 0.800nMAssay Description:Dissociation constant for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKd: 0.200nMAssay Description:Dissociation constant for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Dissociation constant for Retinoid X receptor alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKd: 645nMAssay Description:Dissociation constant for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Dissociation constant for Retinoid X receptor alphaMore data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Dissociation constant for Retinoid X receptor alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKd: >3.00E+4nMAssay Description:Dissociation constant for Retinoic acid receptor gammaMore data for this Ligand-Target Pair