Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 19 hits in this display
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 70.4nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 70.4nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 353nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: >500nMAssay Description:This assay is relatively simple, reasonably sensitive, and the peptide substrate can be adjusted both in terms of sequence and concentration to meet ...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 1.45E+3nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 1.87E+3nMAssay Description:Kinase activity was detected using CisBio HTRF kinEASE kit based on time-resolved fluorescence transfer (FRET). The assay was performed in 384-well w...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 1.87E+3nMAssay Description:RET and KDR: Kinase activity was detected using CisBio HTRF kinEASE kit based on time-resolved fluorescence transfer (FRET). The assay was performed ...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 4.57E+3nMAssay Description:RET and KDR: Kinase activity was detected using CisBio HTRF kinEASE kit based on time-resolved fluorescence transfer (FRET). The assay was performed ...More data for this Ligand-Target Pair
BDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)
IC50: 4.57E+3nMAssay Description:Kinase activity was detected using CisBio HTRF kinEASE kit based on time-resolved fluorescence transfer (FRET). The assay was performed in 384-well w...More data for this Ligand-Target Pair