Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL

LigandBDBM50343659((E)-4-((8-hydroxyquinolin-5-yl)diazenyl)benzoic ac...)Copy SMILESCopy InChI

Affinity DataIC50:  3.47E+3nMAssay Description:Inhibition of RSK2 after 60 minsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetLactoylglutathione lyase(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL

LigandBDBM50343659((E)-4-((8-hydroxyquinolin-5-yl)diazenyl)benzoic ac...)Copy SMILESCopy InChI

Affinity DataIC50:  4.45E+3nMAssay Description:Inhibition of recombinant human N-terminal Met and 6-His-tagged Glyoxalase-1 (Ala2 to Met184 residues) using glutathione and methylglyoxal as substra...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI