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Compile Data Set for Download or QSAR
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Found
9
Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [44-168,333-460]'
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205431
((6S+2S)-PEG1 (7))
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Affinity Data
Ki: 0.0120nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205453
(MTI (35))
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Copy InChI
Affinity Data
Ki: 0.0870nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205435
((6S+2S)-PEG7 (11))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.00590nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205432
((6S+2S)-PEG2 (8))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.00910nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205433
((6S+2S)-PEG3 (9))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.00750nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205434
((6S+2S)-PEG4 (10))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.00660nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205430
((6S+2S)-PEG0 (6))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.0470nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205429
( (R)-JQ1 (3) | US10407441, Compound (R)-JQ1 | US10...)
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Copy InChI
Affinity Data
Kd: 7.30nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Human)
Dana-Farber Cancer Institute
Ligand
BDBM205431
((6S+2S)-PEG1 (7))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.00470nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI