Found 13 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2'
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataIC50: 1.78E+4nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataIC50: 5.23E+4nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataIC50: 4.80E+5nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 690nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile
Curated by ChEMBL
University Of Chile
Curated by ChEMBL
Affinity DataEC50: 790nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair