Affinity DataIC50: 0.0700nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.940nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.29nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair